Pharmacological characterization of AC-90179 [2-(4-methoxyphenyl)-N-(4-methyl-benzyl)-N-(1-methyl-piperidin-4-yl)-acetamide hydrochloride]: a selective serotonin 2A receptor inverse agonist
about
Serotonin, neural markers, and memoryMotoneuron excitability and muscle spasms are regulated by 5-HT2B and 5-HT2C receptor activity.A novel aminotetralin-type serotonin (5-HT) 2C receptor-specific agonist and 5-HT2A competitive antagonist/5-HT2B inverse agonist with preclinical efficacy for psychoses.On the discovery and development of pimavanserin: a novel drug candidate for Parkinson's psychosis.Atypical antipsychotics and inverse agonism at 5-HT2 receptors.Pairings of lever and food induce Pavlovian conditioned approach of sign-tracking and goal-tracking in C57BL/6 mice.5-HT7 receptor activation: procognitive and antiamnesic effects.
P2860
Q26800204-17B589B4-2AB0-4F61-8B56-5407F88D4803Q34686451-708C795A-91F6-492F-B8DA-0F3AC59118EAQ37707718-ECE347BC-BB96-4305-B4F8-DD705D19D4B6Q38200546-A498B3DB-737B-4F5F-B5DD-9EF7D4346F6AQ41250110-5980C95A-BA71-4D6A-B60C-EEFA91035720Q42152825-B8F8D040-AAD6-4678-A27E-CE1AD700C566Q48630264-C5F48F00-8C2C-4893-BDCA-A443F0BFE6F4
P2860
Pharmacological characterization of AC-90179 [2-(4-methoxyphenyl)-N-(4-methyl-benzyl)-N-(1-methyl-piperidin-4-yl)-acetamide hydrochloride]: a selective serotonin 2A receptor inverse agonist
description
2004 nî lūn-bûn
@nan
2004 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
2004 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
2004年の論文
@ja
2004年論文
@yue
2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
@zh-tw
2004年论文
@wuu
name
Pharmacological characterizati ...... in 2A receptor inverse agonist
@ast
Pharmacological characterizati ...... in 2A receptor inverse agonist
@en
Pharmacological characterizati ...... in 2A receptor inverse agonist
@nl
type
label
Pharmacological characterizati ...... in 2A receptor inverse agonist
@ast
Pharmacological characterizati ...... in 2A receptor inverse agonist
@en
Pharmacological characterizati ...... in 2A receptor inverse agonist
@nl
prefLabel
Pharmacological characterizati ...... in 2A receptor inverse agonist
@ast
Pharmacological characterizati ...... in 2A receptor inverse agonist
@en
Pharmacological characterizati ...... in 2A receptor inverse agonist
@nl
P2093
P356
P1476
Pharmacological characterizati ...... in 2A receptor inverse agonist
@en
P2093
Bo-Ragnar Tolf
Carl Magnus Andersson
David M Weiner
Henriette Kold
Isaac Veinbergs
Kimberly E Vanover
Malath Makhay
Mark R Brann
Robert E Davis
Scott C Harvey
P304
P356
10.1124/JPET.104.066688
P407
P577
2004-09-01T00:00:00Z