AM-251 and rimonabant act as direct antagonists at mu-opioid receptors: implications for opioid/cannabinoid interaction studies - sprookjes - yvandenbroek - TriplyDB

AM-251 and rimonabant act as direct antagonists at mu-opioid receptors: implications for opioid/cannabinoid interaction studies

AM-251 and rimonabant act as direct antagonists at mu-opioid receptors: implications for opioid/cannabinoid interaction studies

http://www.wikidata.org/entity/Q28270589

about

Vascular targets for cannabinoids: animal and human studies Tamoxifen Isomers and Metabolites Exhibit Distinct Affinity and Activity at Cannabinoid Receptors: Potential Scaffold for Drug Development Cannabinoid Receptors Are Overexpressed in CLL but of Limited Potential for Therapeutic Exploitation.The Neuroprotective Effect of Lithium in cannabinoid Dependence is Mediated through Modulation of Cyclic AMP, ERK1/2 and GSK-3β Phosphorylation in Cerebellar Granular Neurons of Rat The biarylpyrazole compound AM251 alters mitochondrial physiology via proteolytic degradation of ERRα Self-administration of the anandamide transport inhibitor AM404 by squirrel monkeys Long-term CB₁ receptor blockade enhances vulnerability to anxiogenic-like effects of cannabinoids Elucidating cannabinoid biology in zebrafish (Danio rerio).CB1 and CB2 receptors are novel molecular targets for Tamoxifen and 4OH-Tamoxifen.Selective Estrogen Receptor Modulators: Cannabinoid Receptor Inverse Agonists with Differential CB1 and CB2 Selectivity.Cannabinoids in pain management: CB1, CB2 and non-classic receptor ligands.Characterization of Structurally Novel G Protein Biased CB1 Agonists: Implications for Drug Development.Allostery at opioid receptors: modulation with small molecule ligands.Acetaldehyde as a drug of abuse: insight into AM281 administration on operant-conflict paradigm in rats Antinociceptive effects of the 6-O-sulfate ester of morphine in normal and diabetic rats: Comparative role of mu- and delta-opioid receptors.Characterization of the intrinsic activity for a novel class of cannabinoid receptor ligands: Indole quinuclidine analogs.Exploring the first Rimonabant analog-opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors.Antagonism of cannabinoid receptor 1 attenuates the anti-inflammatory effects of electroacupuncture in a rodent model of migraine.Amphetamine elevates nucleus accumbens dopamine via an action potential-dependent mechanism that is modulated by endocannabinoids.Effects of centrally administered endocannabinoids and opioids on orofacial pain perception in rats.Role of cannabinoid receptor type 1 in tibial and pudendal neuromodulation of bladder overactivity in cats.Genistein Ameliorates Scopolamine-Induced Amnesia in Mice Through the Regulation of the Cholinergic Neurotransmission, Antioxidant System and the ERK/CREB/BDNF Signaling

P2860

Q26862515-0AB5F99D-10F4-41B8-926C-1B358BB4F442 Q28554883-46D3C839-A068-4EFD-A390-4B8AB70BDCE8 Q36036102-BDBDF1BA-BFDE-4EFE-BC90-A528A886078A Q36358395-B8E9F6D8-8C45-49D1-8C64-A1D505AEB48C Q36497790-DF7FFBD6-9995-41DA-A210-488A2175CCAB Q36839896-CB924A69-8AA8-40EA-9989-4357BF100DE5 Q36950835-871E379D-0903-4E01-9A0F-C103C45CCC51 Q37090161-AF2DF1BB-C585-4017-AB9A-B7DBB8E506FD Q37386840-1DB06559-8260-4185-8E1E-3F5F3ED02D7F Q37525458-2320F365-20FE-4D8E-AC2B-9E2FF7F976FF Q38212376-9BE04080-2086-4B28-A2BF-FDC4BC825A6D Q38429080-69C89B20-88F2-4B82-A62E-CDF68170052F Q39248479-2CDF4DDD-F4DC-4616-8358-AC43F079C0C8 Q42060895-694DF67E-9353-48D8-AE08-05B8E0DBA0DF Q42742832-2471A7CD-C9E7-4446-9100-B2856D8AF292 Q43214296-7B0D97BF-7A43-4B2F-BABE-8770388A8F27 Q44342705-AE20BA0D-D0DA-4570-BDDF-64E996840D80 Q47366456-C2D7B1F7-8CC8-46DF-A0BA-4D2F1F877AB5 Q47445865-ED661F7F-D840-4A9A-81B6-1EA894D3D201 Q48298041-CBFF6A36-45B0-4D0A-A10A-D403B44A79C8 Q48403088-9AD5AA92-B39D-4087-A47D-D2AA7134FE5B Q58122657-11557890-0BF7-4BA9-8E3A-E4599EF85FC0

P2860

AM-251 and rimonabant act as direct antagonists at mu-opioid receptors: implications for opioid/cannabinoid interaction studies

http://www.wikidata.org/entity/Q28270589

description

2012 nî lūn-bûn

@nan

2012 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած

@hyw

2012 թվականի հոտեմբերին հրատարակված գիտական հոդված

@hy

2012年の論文

@ja

2012年論文

@yue

2012年論文

@zh-hant

2012年論文

@zh-hk

2012年論文

@zh-mo

2012年論文

@zh-tw

2012年论文

@wuu

name

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@ast

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@en

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@nl

type

label

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@ast

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@en

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@nl

prefLabel

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@ast

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@en

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@nl

P1433

Q28270589-CFDE4C0E-6C3C-4A98-9789-F3BBD95074B2

P1476

Q28270589-003F8129-51C3-4C49-BA2C-D8784484066D

P2093

Q28270589-2759ADF6-A375-4AE1-B22F-5E4C125C9444

Q28270589-433AB84D-9673-4F0A-8C8E-7B28E6EE15CF

Q28270589-76DA85E8-B9FE-4FA7-ADBB-4FA68E9766A0

Q28270589-C67CDC45-1AA5-40AC-8634-90B3F11F7872

Q28270589-D0898AF7-0BDA-42E1-8553-F300003A124D

Q28270589-D3384F96-1BB7-4B52-86AA-F3148B74DA63

Q28270589-D5B851DF-CFA2-415D-A423-98BED6353383

P2860

Q28270589-02623AD6-F1F7-4DE3-9A81-3772F4B6612E

Q28270589-04B20BBA-5630-4F0F-848B-F76F2A46371C

Q28270589-0A43862D-19A4-4B76-A891-A5BB99ED3B6C

Q28270589-0CFFE522-F794-4528-99C5-7FAF01D4A5C2

Q28270589-1199C984-466D-49F6-B81F-49DBEC49DF6B

Q28270589-13BDBD24-610C-4AA5-9D0F-9E6DBE19214B

Q28270589-154FA45B-5E6B-485C-A6C5-58AF98A77261

Q28270589-1940C69D-A2C0-463F-BAF7-9E4056346506

Q28270589-1D702740-EF47-4726-A507-BF053632D059

Q28270589-2C3DB2B9-D89B-4B2A-98AC-B411D1F7403E

P304

Q28270589-59B576D1-CFF9-4A44-993F-540D14D7BEA4

P31

Q28270589-20780926-269F-4D49-A031-4EAC64A2D679

P3181

Q28270589-EA6EB893-6F7F-4CD5-8CCA-3A7DF8163B2F

P356

Q28270589-206D6935-6A6D-4E61-8444-88189C7FE399

P407

Q28270589-58491130-F790-4145-86C5-63073A8DCBF1

P433

Q28270589-08569C3E-AB5B-4594-8FE3-C1F43068C30B

P478

Q28270589-B83F7322-8D06-4A71-B234-A5FF0CB40DF9

P577

Q28270589-EAB23D42-F75D-485F-BF86-6B79AA93C01E

P698

Q28270589-5CADA2BB-3C1E-4ED8-8D40-0181FC560361

P921

Q28270589-6E3DCFD5-FBA3-486E-B0E0-CB6D90A20D9C

Q28270589-B0473FA7-2652-4187-A218-3D863F886F2C

Q28270589-C048BE6C-9613-4428-A048-A89672CE087D

Q28270589-f9f635b5-75fd-4398-bbf9-bbcdc065f805

P932

Q28270589-0246669A-809B-4625-B3E0-29D90CC83F0C

P3181

P356

J.NEUROPHARM.2012.06.046

P1433

Neuropharmacology

P1476

AM-251 and rimonabant act as d ...... annabinoid interaction studies

@en

P2093

Kathryn A Seely

http://www.w3.org/2001/XMLSchema#string

Lirit N Franks

http://www.w3.org/2001/XMLSchema#string

Lisa K Brents

http://www.w3.org/2001/XMLSchema#string

Maheswari Rajasekaran

http://www.w3.org/2001/XMLSchema#string

Paul L Prather

http://www.w3.org/2001/XMLSchema#string

Sarah M Zimmerman

http://www.w3.org/2001/XMLSchema#string

William E Fantegrossi

http://www.w3.org/2001/XMLSchema#string

P2860

Phase I hydroxylated metabolites of the K2 synthetic cannabinoid JWH-018 retain in vitro and in vivo cannabinoid 1 receptor affinity and activity

Evidence that the plant cannabinoid Delta9-tetrahydrocannabivarin is a cannabinoid CB1 and CB2 receptor antagonist

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

The endocannabinoid noladin ether acts as a full agonist at human CB2 cannabinoid receptors

Activation of mitogen-activated protein kinases by stimulation of the central cannabinoid receptor CB1

Signaling pathway associated with stimulation of CB2 peripheral cannabinoid receptor. Involvement of both mitogen-activated protein kinase and induction of Krox-24 expression

Therapeutic potential of cannabis in pain medicine

Comparison of the pharmacology and signal transduction of the human cannabinoid CB1 and CB2 receptors

Immune regulation by cannabinoid compounds through the inhibition of the cyclic AMP signaling cascade and altered gene expression

Structure-activity relationships of pyrazole derivatives as cannabinoid receptor antagonists

P304

905-15

http://www.w3.org/2001/XMLSchema#string

P31

scholarly article

P3181

1116023

http://www.w3.org/2001/XMLSchema#string

P356

10.1016/J.NEUROPHARM.2012.06.046

http://www.w3.org/2001/XMLSchema#string

P407

P433

5

http://www.w3.org/2001/XMLSchema#string

P478

63

http://www.w3.org/2001/XMLSchema#string

P577

2012-10-01T00:00:00Z

http://www.w3.org/2001/XMLSchema#dateTime

P698

22771770

http://www.w3.org/2001/XMLSchema#string

P921

cannabinoid receptor

P932

3408547

http://www.w3.org/2001/XMLSchema#string