Ion Channel Blockers as Antimicrobial Agents, Efflux Inhibitors, and Enhancers of Macrophage Killing Activity against Drug Resistant Mycobacterium tuberculosis
about
Interplay between Mutations and Efflux in Drug Resistant Clinical Isolates of Mycobacterium tuberculosisMode of action of the 2-phenylquinoline efflux inhibitor PQQ4R against Escherichia coli.Thioridazine: A Non-Antibiotic Drug Highly Effective, in Combination with First Line Anti-Tuberculosis Drugs, against Any Form of Antibiotic Resistance of Mycobacterium tuberculosis Due to Its Multi-Mechanisms of Action.Targeting Energy Metabolism in Mycobacterium tuberculosis, a New Paradigm in Antimycobacterial Drug Discovery.Analogues of Disulfides from Allium stipitatum Demonstrate Potent Anti-tubercular Activities through Drug Efflux Pump and Biofilm Inhibition.Combined chemical genetics and data-driven bioinformatics approach identifies receptor tyrosine kinase inhibitors as host-directed antimicrobials.Efflux Activity Differentially Modulates the Levels of Isoniazid and Rifampicin Resistance among Multidrug Resistant and Monoresistant Mycobacterium tuberculosis Strains.Identification of a Novel Polyamine Scaffold With Potent Efflux Pump Inhibition Activity Toward Multi-Drug Resistant Bacterial Pathogens.Challenging the Drug-Likeness Dogma for New Drug Discovery in Tuberculosis
P2860
Q33607162-0190AEB9-B9FC-4C35-9862-B58498B285EAQ38682599-B34A446E-764B-4815-B030-173716A2C4FDQ38872058-629021A9-3820-4F79-8526-44523A2CADE4Q39235946-3837064B-8639-448C-B884-F88538D70A07Q47710524-EA341002-FC3A-4120-9B75-E06B38016531Q48171420-89F9D588-A90B-47B0-89FB-9189F02ABBDEQ53704257-E33C19D7-45B9-4327-96C1-5AA77F469E34Q55398494-9C7D33BD-CF3E-4625-881F-73DC1F420B2EQ57656314-338310C2-BA09-43B7-ABB2-140C7A13F247
P2860
Ion Channel Blockers as Antimicrobial Agents, Efflux Inhibitors, and Enhancers of Macrophage Killing Activity against Drug Resistant Mycobacterium tuberculosis
description
2016 nî lūn-bûn
@nan
2016 թուականին հրատարակուած գիտական յօդուած
@hyw
2016 թվականին հրատարակված գիտական հոդված
@hy
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
name
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@ast
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@en
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@nl
type
label
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@ast
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@en
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@nl
prefLabel
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@ast
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@en
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@nl
P2860
P50
P921
P1433
P1476
Ion Channel Blockers as Antimi ...... ant Mycobacterium tuberculosis
@en
P2860
P304
P356
10.1371/JOURNAL.PONE.0149326
P407
P50
P577
2016-01-01T00:00:00Z