Combinatorial compound libraries for drug discovery: an ongoing challenge.
about
When Quality Beats Quantity: Decision Theory, Drug Discovery, and the Reproducibility CrisisDiscovery of active proteins directly from combinatorial randomized protein libraries without display, purification or sequencing: identification of novel zinc finger proteinsIdentifying the immunomodulatory components of helminthsStructural Analysis of Charge Discrimination in the Binding of Inhibitors to Human Carbonic Anhydrases I and IIPhage protein-targeted cancer nanomedicines.Microengineering methods for cell-based microarrays and high-throughput drug-screening applicationsDocking challenge: protein sampling and molecular docking performance.Estimation of the size of drug-like chemical space based on GDB-17 data.Automated ARGET ATRP Accelerates Catalyst Optimization for the Synthesis of Thiol-Functionalized Polymers.Fluorous-enhanced multicomponent reactions for making drug-like library scaffolds.Microwave-Enhanced High-Speed Fluorous Synthesis.Development of a fluorescence-based, ultra high-throughput screening platform for nanoliter-scale cytochrome p450 microarrays.Mutations in fd phage major coat protein modulate affinity of the displayed peptideHigh-throughput in vivo screening of targeted molecular imaging agents.'On-the-fly' optical encoding of combinatorial peptide libraries for profiling of protease specificity.The Privileged Chemical Space Predictor (PCSP): a computer program that identifies privileged chemical space from screens of modularly assembled chemical libraries.A peptide & peptide nucleic acid synthesis technology for transporter molecules and theranostics--the SPPS.A sandwiched microarray platform for benchtop cell-based high throughput screening.Metabolizing enzyme toxicology assay chip (MetaChip) for high-throughput microscale toxicity analyses.High-throughput small molecule identification using MALDI-TOF and a nanolayered substrate.Microwave-assisted tandem transformation on an ionic-liquid support: efficient synthesis of pyrrolo/pyridobenzimidazolones and isoindolinone-fused benzimidazoles.Combinatorial synthesis of chemically diverse core-shell nanoparticles for intracellular delivery.Photo-assisted peptide enrichment in protein complex cross-linking analysis of a model homodimeric protein using mass spectrometry.Protein denaturation and protein:drugs interactions from intrinsic protein fluorescence measurements at the nanolitre scaleHigh-throughput enzyme assay on a multichannel microchip using optically gated sample introductionMicrowave and continuous flow technologies in drug discovery.Towards microfluidic technology-based MALDI-MS platforms for drug discovery: a review.Biomedical engineering strategies in system design space.Solution-phase parallel synthesis of acyclic nucleoside libraries of purine, pyrimidine, and triazole acetamides.Drug discovery in academia.Incorporating Virtual Reactions into a Logic-based Ligand-based Virtual Screening Method to Discover New LeadsA New Application of Parallel Synthesis Strategy for Discovery of Amide-Linked Small Molecules as Potent Chondroprotective Agents in TNF-α-Stimulated Chondrocytes.Screening of Small Molecule Microarrays for Ligands Targeted to the Extracellular Epitopes of Living Cells.Three-dimensional cellular microarray for high-throughput toxicology assaysControl and detection of chemical reactions in microfluidic systems.High-throughput cellular microarray platforms: applications in drug discovery, toxicology and stem cell researchSystematizing serendipity for cardiovascular drug discovery.Molecules that modulate Apaf-1 activity.Advances in cell-based biosensors using three-dimensional cell-encapsulating hydrogels.Action of natural products on p2 receptors: a reinvented era for drug discovery.
P2860
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P2860
Combinatorial compound libraries for drug discovery: an ongoing challenge.
description
2003 nî lūn-bûn
@nan
2003 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
2003 թվականի մարտին հրատարակված գիտական հոդված
@hy
2003年の論文
@ja
2003年論文
@yue
2003年論文
@zh-hant
2003年論文
@zh-hk
2003年論文
@zh-mo
2003年論文
@zh-tw
2003年论文
@wuu
name
Combinatorial compound libraries for drug discovery: an ongoing challenge.
@ast
Combinatorial compound libraries for drug discovery: an ongoing challenge.
@en
type
label
Combinatorial compound libraries for drug discovery: an ongoing challenge.
@ast
Combinatorial compound libraries for drug discovery: an ongoing challenge.
@en
prefLabel
Combinatorial compound libraries for drug discovery: an ongoing challenge.
@ast
Combinatorial compound libraries for drug discovery: an ongoing challenge.
@en
P2093
P2860
P356
P1476
Combinatorial compound libraries for drug discovery: an ongoing challenge.
@en
P2093
David Wagner
Frank Schoenen
H Mario Geysen
Richard Wagner
P2860
P2888
P304
P356
10.1038/NRD1035
P577
2003-03-01T00:00:00Z