about
Structure-based design, synthesis, and biochemical and pharmacological characterization of novel salvinorin A analogues as active state probes of the kappa-opioid receptorThe effects of herkinorin, the first mu-selective ligand from a salvinorin A-derived scaffold, in a neuroendocrine biomarker assay in nonhuman primatesKappa-opioid ligands in the study and treatment of mood disordersCollybolide is a novel biased agonist of κ-opioid receptors with potent antipruritic activityNeuropharmacology of the naturally occurring kappa-opioid hallucinogen salvinorin AChemical methods for the synthesis and modification of neoclerodane diterpenesSalvinorin A analogs and other κ-opioid receptor compounds as treatments for cocaine abuse.Effect of kappa-opioid receptor agonists U69593, U50488H, spiradoline and salvinorin A on cocaine-induced drug-seeking in rats.Opioid receptor probes derived from cycloaddition of the hallucinogen natural product salvinorin A.Pharmacology and anti-addiction effects of the novel κ opioid receptor agonist Mesyl Sal B, a potent and long-acting analogue of salvinorin ASynthesis and biological evaluation of C-2 halogenated analogs of salvinorin A.Salvinorin A and derivatives: protection from metabolism does not prolong short-term, whole-brain residence.Natural products as tools for neuroscience: discovery and development of novel agents to treat drug abuseSynthetic studies of neoclerodane diterpenoids from Salvia splendens and evaluation of Opioid Receptor affinity.The 2-methoxy methyl analogue of salvinorin A attenuates cocaine-induced drug seeking and sucrose reinforcements in rats.Palladium-catalyzed transformations of salvinorin A, a neoclerodane diterpene from Salvia divinorum.Utilizing nature as a source of new probes for opioid pharmacology.Clerodane diterpenes: sources, structures, and biological activities.Modification of the furan ring of salvinorin A: identification of a selective partial agonist at the kappa opioid receptor.Novel neoclerodane diterpene derivatives from the smoke of salvinorin A.Synergistic blockade of alcohol escalation drinking in mice by a combination of novel kappa opioid receptor agonist Mesyl Salvinorin B and naltrexone.Addressing Structural Flexibility at the A-Ring on Salvinorin A: Discovery of a Potent Kappa-Opioid Agonist with Enhanced Metabolic Stability.Semisynthesis and Kappa-Opioid Receptor Activity of Derivatives of Columbin, a Furanolactone Diterpene.Dynamic Strategic Bond Analysis Yields a Ten-Step Synthesis of 20-nor-Salvinorin A, a Potent κ-OR Agonist.Total Synthesis of (-)-Salvinorin A.O6C-20-nor-salvinorin A is a stable and potent KOR agonist.
P2860
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P2860
description
2008 nî lūn-bûn
@nan
2008 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Salvinorin A analogs as probes in opioid pharmacology.
@ast
Salvinorin A analogs as probes in opioid pharmacology.
@en
type
label
Salvinorin A analogs as probes in opioid pharmacology.
@ast
Salvinorin A analogs as probes in opioid pharmacology.
@en
prefLabel
Salvinorin A analogs as probes in opioid pharmacology.
@ast
Salvinorin A analogs as probes in opioid pharmacology.
@en
P2860
P356
P1433
P1476
Salvinorin A analogs as probes in opioid pharmacology.
@en
P2093
Richard B Rothman
Thomas E Prisinzano
P2860
P304
P356
10.1021/CR0782269
P577
2008-05-01T00:00:00Z