Compounds that activate the mouse melanocortin-1 receptor identified by screening a small molecule library based upon the beta-turn.
about
Synthesis of dimeric trifluoromethoxyacridine-derived pathogen-inactivating nucleic acid intercalators.Ligand-based peptide design and combinatorial peptide libraries to target G protein-coupled receptorsPrivileged diazepine compounds and their emergence as bromodomain inhibitors.Peptide interactions with G-protein coupled receptors.Privileged scaffolds targeting reverse-turn and helix recognition.Pharmacologic induction of epidermal melanin and protection against sunburn in a humanized mouse model.Bench-top to clinical therapies: A review of melanocortin ligands from 1954 to 2016.Modified melanocortin tetrapeptide Ac-His-dPhe-Arg-Trp-NH at the arginine side chain with ureas and thioureas.Beta-turn secondary structure and melanocortin ligands.Semi-rigid tripeptide agonists of melanocortin receptors.Structure-activity studies on the corticotropin releasing factor antagonist astressin, leading to a minimal sequence necessary for antagonistic activity.Ester vs. amide on folding: a case study with a 2-residue synthetic peptide.Synthesis and Structure-Activity Relationships of Substituted Urea Derivatives on Mouse Melanocortin Receptors.Cyclopropane-Based Peptidomimetics Mimicking Wide-Ranging Secondary Structures of Peptides: Conformational Analysis and Their Use in Rational Ligand Optimization.From Peptides to Peptidomimetics: A Strategy Based on the Structural Features of Cyclopropane.
P2860
Q30320423-C72491F3-A959-4398-9658-5A17FE523F40Q33650270-4C125C59-9966-4FF0-A5C6-8A9F8671B5ECQ33671341-F69D0997-8963-4CD9-8379-6FA5E447AE79Q34483031-A450A949-FFC1-4D1A-82AB-CBDCD70EC61DQ37030888-CDB0AF59-5EDC-44DF-871C-74726BE22D92Q37380135-0A856A3D-80A9-4E03-A01C-8A25734DF778Q39211934-7D63996D-F1B9-4B72-8251-054C1E2153CCQ40363165-20A7C4D9-2023-48B9-9E43-1E53A071207EQ41957100-B61E07FC-C9ED-4971-9E1E-55F5045F78EDQ41962062-73A842AE-2B2E-46B1-A81D-F27DA561A27BQ44784411-CAFE8C45-C564-4A79-9F32-09E6B6418368Q45329378-4F9ABB3D-2CCD-4E31-8DE9-10ADB490B034Q47120733-4BEDF4CA-AAB3-4E5F-A0E5-ED6100BA3E11Q48130657-FEC7520D-CF9D-43ED-BA67-67E2654F4B83Q48250705-4B9AC64B-EBEF-4A7A-9308-10EA9A3FF845
P2860
Compounds that activate the mouse melanocortin-1 receptor identified by screening a small molecule library based upon the beta-turn.
description
1999 nî lūn-bûn
@nan
1999 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1999 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
1999年の論文
@ja
1999年論文
@yue
1999年論文
@zh-hant
1999年論文
@zh-hk
1999年論文
@zh-mo
1999年論文
@zh-tw
1999年论文
@wuu
name
Compounds that activate the mo ...... rary based upon the beta-turn.
@ast
Compounds that activate the mo ...... rary based upon the beta-turn.
@en
type
label
Compounds that activate the mo ...... rary based upon the beta-turn.
@ast
Compounds that activate the mo ...... rary based upon the beta-turn.
@en
prefLabel
Compounds that activate the mo ...... rary based upon the beta-turn.
@ast
Compounds that activate the mo ...... rary based upon the beta-turn.
@en
P2093
P356
P1476
Compounds that activate the mo ...... rary based upon the beta-turn.
@en
P2093
Haskell-Luevano C
Rosenquist A
P304
P356
10.1021/JM990190S
P407
P577
1999-10-01T00:00:00Z