Molecular basis of pimarane compounds as novel activators of large-conductance Ca(2+)-activated K(+) channel alpha-subunit.
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The intermediate-conductance calcium-activated potassium channel KCa3.1 contributes to atherogenesis in mice and humansOn benzofuroindole analogues as smooth muscle relaxantsDirect synthesis of Z-alkenyl halides through catalytic cross-metathesisA protective mechanism against antibiotic-induced ototoxicity: role of prestinResin-acid derivatives as potent electrostatic openers of voltage-gated K channels and suppressors of neuronal excitabilityNatural products that reduce rotavirus infectivity identified by a cell-based moderate-throughput screening assay1,4a,7-Trimethyl-7-vinyl-1,2,3,4,4a,4b,5,6,7,9,10,10a-dodeca-hydro-phenanthrene-1-carboxylic acid.Calcium- and voltage-gated potassium (BK) channel activators in the 5β-cholanic acid-3α-ol analogue series with modifications in the lateral chainKinetically controlled E-selective catalytic olefin metathesis.Resin acid conversion with CYP105A1: an enzyme with potential for the production of pharmaceutically relevant diterpenoids.Effects of the novel BK (KCa 1.1) channel opener GoSlo-SR-5-130 are dependent on the presence of BKβ subunits.Synergistic antinociception by the cannabinoid receptor agonist anandamide and the PPAR-alpha receptor agonist GW7647.Modulation by simvastatin of iberiotoxin-sensitive, Ca2+-activated K+ channels of porcine coronary artery smooth muscle cells.K+ channel modulators for the treatment of neurological disorders and autoimmune diseasesInhibition of vascular calcium-gated chloride currents by blockers of KCa1.1, but not by modulators of KCa2.1 or KCa2.3 channels.Ginsenoside Rg3 enhances large conductance Ca2+-activated potassium channel currents: a role of Tyr360 residue.Drug-induced ion channel opening tuned by the voltage sensor charge profile.Isopimaric acid - a multi-targeting ion channel modulator reducing excitability and arrhythmicity in a spontaneously beating mouse atrial cell line.A large-conductance (BK) potassium channel subtype affects both growth and mineralization of human osteoblasts.Activation of large-conductance, Ca2+-activated K+ channels by cannabinoids.Synthetic Studies on Tricyclic Diterpenoids: Direct Allylic Amination Reaction of Isopimaric Acid DerivativesCalcium-activated and voltage-gated potassium channels of the pancreatic islet impart distinct and complementary roles during secretagogue induced electrical responses.Stereoselective Carbonyl Olefination with Fluorosulfoximines: Facile Access to Z or E Terminal Monofluoroalkenes.Calcineurin inhibitors suppress the high-temperature stress sensitivity of the yeast ubiquitin ligase Rsp5 mutant: a new method of screening for calcineurin inhibitors.Atom-by-atom tuning of the electrostatic potassium-channel modulator dehydroabietic acid.
P2860
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P2860
Molecular basis of pimarane compounds as novel activators of large-conductance Ca(2+)-activated K(+) channel alpha-subunit.
description
2002 nî lūn-bûn
@nan
2002 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2002 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2002年の論文
@ja
2002年論文
@yue
2002年論文
@zh-hant
2002年論文
@zh-hk
2002年論文
@zh-mo
2002年論文
@zh-tw
2002年论文
@wuu
name
Molecular basis of pimarane compounds as novel activators of large-conductance Ca
@nl
Molecular basis of pimarane co ...... ed K(+) channel alpha-subunit.
@ast
Molecular basis of pimarane co ...... ed K(+) channel alpha-subunit.
@en
type
label
Molecular basis of pimarane compounds as novel activators of large-conductance Ca
@nl
Molecular basis of pimarane co ...... ed K(+) channel alpha-subunit.
@ast
Molecular basis of pimarane co ...... ed K(+) channel alpha-subunit.
@en
prefLabel
Molecular basis of pimarane compounds as novel activators of large-conductance Ca
@nl
Molecular basis of pimarane co ...... ed K(+) channel alpha-subunit.
@ast
Molecular basis of pimarane co ...... ed K(+) channel alpha-subunit.
@en
P2093
P356
P1476
Molecular basis of pimarane co ...... ed K(+) channel alpha-subunit.
@en
P2093
Aki Yamada
Katsuhiko Muraki
Kazuho Sakamoto
Masanobu Uchiyama
Susumu Ohya
Tomohiko Ohwada
Yuji Imaizumi
P304
P356
10.1124/MOL.62.4.836
P577
2002-10-01T00:00:00Z