Determinants of activity at human Toll-like receptors 7 and 8: quantitative structure-activity relationship (QSAR) of diverse heterocyclic scaffolds.
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Comparative Geometrical Analysis of Leucine-Rich Repeat Structures in the Nod-Like and Toll-Like Receptors in Vertebrate Innate Immunity.Virtual Screening Approaches towards the Discovery of Toll-Like Receptor ModulatorsIdentification of Adjuvantic Activity of Amphotericin B in a Novel, Multiplexed, Poly-TLR/NLR High-Throughput Screen.Enrichment assessment of multiple virtual screening strategies for Toll-like receptor 8 agonists based on a maximal unbiased benchmarking data set.The Imidazoquinoline Toll-Like Receptor-7/8 Agonist Hybrid-2 Potently Induces Cytokine Production by Human Newborn and Adult Leukocytes.Structure-Based Design of Human TLR8-Specific Agonists with Augmented Potency and Adjuvanticity.Insights on the mechanism of action of immunostimulants in relation to their pharmacological potency. The effects of imidazoquinolines on TLR8.Structural aspects of nucleic acid-sensing Toll-like receptors.Toward a structural understanding of nucleic acid-sensing Toll-like receptors in the innate immune system.Development of a web-based platform for studying lithiation reactions in silico.Cascade bicyclization of triethylammonium thiolates with hydrazines: efficient access to pyrazolo[3,4-c]quinolines.Protamine-stabilized RNA as an ex vivo stimulant of primary human dendritic cell subsets.Syntheses of Human TLR8-Specific Small-Molecule Agonists.
P2860
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P2860
Determinants of activity at human Toll-like receptors 7 and 8: quantitative structure-activity relationship (QSAR) of diverse heterocyclic scaffolds.
description
2014 nî lūn-bûn
@nan
2014 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
Determinants of activity at hu ...... iverse heterocyclic scaffolds.
@ast
Determinants of activity at hu ...... iverse heterocyclic scaffolds.
@en
Determinants of activity at hu ...... tructure-activity relationship
@nl
type
label
Determinants of activity at hu ...... iverse heterocyclic scaffolds.
@ast
Determinants of activity at hu ...... iverse heterocyclic scaffolds.
@en
Determinants of activity at hu ...... tructure-activity relationship
@nl
prefLabel
Determinants of activity at hu ...... iverse heterocyclic scaffolds.
@ast
Determinants of activity at hu ...... iverse heterocyclic scaffolds.
@en
Determinants of activity at hu ...... tructure-activity relationship
@nl
P2093
P2860
P50
P356
P1476
Determinants of activity at hu ...... iverse heterocyclic scaffolds.
@en
P2093
Alec R Hermanson
Alex C D Salyer
Hiromi Tanji
Manoj Kumar
Rajalakshmi Balakrishna
Subbalakshmi S Malladi
Sunil A David
Toshiyuki Shimizu
Umeharu Ohto
P2860
P304
P356
10.1021/JM500744F
P407
P577
2014-09-17T00:00:00Z