Identification and characterization of inhibitors of bacterial enoyl-acyl carrier protein reductase - sprookjes - yvandenbroek - TriplyDB

Identification and characterization of inhibitors of bacterial enoyl-acyl carrier protein reductase

Identification and characterization of inhibitors of bacterial enoyl-acyl carrier protein reductase

http://www.wikidata.org/entity/Q34315832

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Crystal structure of enoyl-acyl carrier protein reductase (FabK) fromStreptococcus pneumoniaereveals the binding mode of an inhibitor Structural and Enzymatic Analyses Reveal the Binding Mode of a Novel Series of Francisella tularensis Enoyl Reductase (FabI) Inhibitors Mechanism and inhibition of saFabI, the enoyl reductase from Staphylococcus aureus Challenges of antibacterial discovery The MUT056399 inhibitor of FabI is a new antistaphylococcal compound.In silico target fishing and pharmacological profiling for the isoquinoline alkaloids of Macleaya cordata (Bo Luo Hui)Inhibiting bacterial fatty acid synthesis.The application of Tet repressor in prokaryotic gene regulation and expression Enoyl acyl carrier protein reductase inhibitors: a patent review (2006 - 2010).Recent advances in inhibitors of bacterial fatty acid synthesis type II (FASII) system enzymes as potential antibacterial agents.Crystallization and preliminary X-ray crystallographic analysis of enoyl-ACP reductase III (FabL) from Bacillus subtilis.Studies of Staphylococcus aureus FabI inhibitors: fragment-based approach based on holographic structure-activity relationship analyses.Crystallization and preliminary X-ray analysis of enoyl-acyl carrier protein reductase (FabK) from Streptococcus pneumoniae New 2-thiopyridines as potential candidates for killing both actively growing and dormant Mycobacterium tuberculosis cells.Purification, crystallization and preliminary X-ray diffraction analysis of enoyl-acyl carrier protein reductase (FabK) from Streptococcus mutans strain UA159 AG205, a novel agent directed against FabK of Streptococcus pneumoniae.Pharmacophore and molecular docking guided 3D-QSAR study of bacterial enoyl-ACP reductase (FabI) Inhibitors.Utilization of target-specific, hypersensitive strains of Saccharomyces cerevisiae to determine the mode of action of antifungal compounds.3D-QSAR studies on triclosan derivatives as Plasmodium falciparum enoyl acyl carrier reductase inhibitors.Molecular modeling studies and anti-TB activity of trisubstituted indolizine analogues; molecular docking and dynamic inputs.Rational questing for potential novel inhibitors of FabK from Streptococcus pneumoniae by combining FMO calculation, CoMFA 3D-QSAR modeling and virtual screening.Macromolecular synthesis and membrane perturbation assays for mechanisms of action studies of antimicrobial agents.

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Identification and characterization of inhibitors of bacterial enoyl-acyl carrier protein reductase

http://www.wikidata.org/entity/Q34315832

description

2004 nî lūn-bûn

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2004 թուականի Մայիսին հրատարակուած գիտական յօդուած

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2004 թվականի մայիսին հրատարակված գիտական հոդված

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2004年の論文

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2004年論文

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2004年論文

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2004年論文

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2004年論文

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2004年論文

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2004年论文

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name

Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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Identification and characteriz ...... acyl carrier protein reductase

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AAC.48.5.1541-1547.2004

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Antimicrobial Agents and Chemotherapy

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Identification and characteriz ...... acyl carrier protein reductase

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Anthony C Arvanites

http://www.w3.org/2001/XMLSchema#string

Bolin Geng

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Debra M Mills

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Donald T Moir

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Gilles Carmel

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Hernan Orgueira

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Jun Fan

http://www.w3.org/2001/XMLSchema#string

Jun Xian

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Losee L Ling

http://www.w3.org/2001/XMLSchema#string

Mark A Ashwell

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P2860

Molecular basis of triclosan activity

Crystal structure of the bacterial membrane protein TolC central to multidrug efflux and protein export

1,4-Disubstituted imidazoles are potential antibacterial agents functioning as inhibitors of enoyl acyl carrier protein reductase (FabI)

Inhibitors of bacterial enoyl acyl carrier protein reductase (FabI): 2,9-disubstituted 1,2,3,4-tetrahydropyrido[3,4-b]indoles as potential antibacterial agents

Discovery of aminopyridine-based inhibitors of bacterial enoyl-ACP reductase (FabI)

A Simple Statistical Parameter for Use in Evaluation and Validation of High Throughput Screening Assays

Whole genome sequencing of meticillin-resistant Staphylococcus aureus

Enzymatic characterization of the target for isoniazid in Mycobacterium tuberculosis

The enoyl-[acyl-carrier-protein] reductases FabI and FabL from Bacillus subtilis

An array of target-specific screening strains for antibacterial discovery.

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1541-1547

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scholarly article

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10.1128/AAC.48.5.1541-1547.2004

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5

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48

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2004-05-01T00:00:00Z

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8600018

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