about
PfCRT and its role in antimalarial drug resistanceFunctional characterization of the Plasmodium falciparum chloroquine-resistance transporter (PfCRT) in transformed Dictyostelium discoideum vesiclesA process similar to autophagy is associated with cytocidal chloroquine resistance in Plasmodium falciparumEvolution of Fitness Cost-Neutral Mutant PfCRT Conferring P. falciparum 4-Aminoquinoline Drug Resistance Is Accompanied by Altered Parasite Metabolism and Digestive Vacuole PhysiologyFusion of field studies and the laboratory solves a puzzle in antimalarial resistanceSecond generation steroidal 4-aminoquinolines are potent, dual-target inhibitors of the botulinum neurotoxin serotype A metalloprotease and P. falciparum malariaRuthenium(II) arene complexes with chelating chloroquine analogue ligands: synthesis, characterization and in vitro antimalarial activity.Plasmodium drug targets outside the genetic control of the parasite.Antiplasmodial activity of chloroquine analogs against chloroquine-resistant parasites, docking studies and mechanisms of drug actionPlasmodium falciparum resistance to cytocidal versus cytostatic effects of chloroquine.Analysis of chloroquine resistance transporter (CRT) isoforms and orthologues in S. cerevisiae yeastPlasmodium falciparum chloroquine resistance transporter is a H+-coupled polyspecific nutrient and drug exporter.Reversed chloroquine molecules as a strategy to overcome resistance in malaria.Chloroquine sensitivity: diminished prevalence of chloroquine-resistant gene marker pfcrt-76 13 years after cessation of chloroquine use in Msambweni, KenyaSontochin as a guide to the development of drugs against chloroquine-resistant malaria.Tricks in Plasmodium's molecular repertoire--escaping 3'UTR excision-based conditional silencing of the chloroquine resistance transporter gene.Combinatorial Genetic Modeling of pfcrt-Mediated Drug Resistance Evolution in Plasmodium falciparum.Globally prevalent PfMDR1 mutations modulate Plasmodium falciparum susceptibility to artemisinin-based combination therapies.Functional Comparison of 45 Naturally Occurring Isoforms of the Plasmodium falciparum Chloroquine Resistance Transporter (PfCRT).Dual-functioning antimalarials that inhibit the chloroquine-resistance transporter."Drug resistance associated membrane proteins".To kill or not to kill, that is the question: cytocidal antimalarial drug resistance.Plasmodium falciparum chloroquine resistance transporter (PfCRT) isoforms PH1 and PH2 perturb vacuolar physiology.Deciphering the Resistance-Counteracting Functions of Ferroquine in Plasmodium falciparum-Infected Erythrocytes.Function of resistance conferring Plasmodium falciparum chloroquine resistance transporter isoforms.Cytostatic versus cytocidal activities of chloroquine analogues and inhibition of hemozoin crystal growth.Relative to quinine and quinidine, their 9-epimers exhibit decreased cytostatic activity and altered heme binding but similar cytocidal activity versus Plasmodium falciparum.Imported and autochthonous malaria in West Saudi Arabia: results from a reference hospital
P2860
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P2860
description
2010 nî lūn-bûn
@nan
2010 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
PfCRT-mediated drug transport in malarial parasites.
@ast
PfCRT-mediated drug transport in malarial parasites.
@en
type
label
PfCRT-mediated drug transport in malarial parasites.
@ast
PfCRT-mediated drug transport in malarial parasites.
@en
prefLabel
PfCRT-mediated drug transport in malarial parasites.
@ast
PfCRT-mediated drug transport in malarial parasites.
@en
P2860
P356
P1433
P1476
PfCRT-mediated drug transport in malarial parasites.
@en
P2093
Paul D Roepe
P2860
P304
P356
10.1021/BI101638N
P407
P577
2010-12-22T00:00:00Z