Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
about
A Novel Allosteric Activator of Free Fatty Acid 2 Receptor Displays Unique Gi-functional BiasCarbetocin is a Functional Selective Gq Agonist That Does Not Promote Oxytocin Receptor Recycling After Inducing β-Arrestin-Independent InternalisationEvolutionary and Comparative Genomics to Drive Rational Drug Design, with Particular Focus on Neuropeptide Seven-Transmembrane Receptors.From Belly to Brain: Targeting the Ghrelin Receptor in Appetite and Food Intake Regulation.Development of Fluorinated Non-Peptidic Ghrelin Receptor Ligands for Potential Use in Molecular Imaging.G protein stoichiometry dictates biased agonism through distinct receptor-G protein partitioning.GHSR-D2R heteromerization modulates dopamine signaling through an effect on G protein conformation.Conditional and Reversible Activation of Class A and B G Protein-Coupled Receptors Using Tethered Pharmacology.Quinolones Modulate Ghrelin Receptor Signaling: Potential for a Novel Small Molecule Scaffold in the Treatment of Cachexia.Selective homodimerization of unprotected peptides using hybrid hydroxydimethylsilane derivativesMaking Sense of Pharmacology: Inverse Agonism and Functional SelectivityGhrelin Receptor Antagonism of Methamphetamine-Induced Conditioned Place Preference and Intravenous Self-Administration in Rats
P2860
Q37227642-CA3B3715-B235-491C-AA46-156097D3BCB2Q37252520-45963A89-B50C-474F-A42A-8CBB157C9AD6Q37551922-B7FF0C95-1D1A-491E-B450-EFA6251CF77AQ37690695-EAE94AC3-5525-46A7-B075-C938F5E0568DQ38734724-74425D8B-03CE-489B-B145-FE968F208CE8Q41367745-820ED81A-FA70-498C-B71C-8E3D50092775Q52327561-49EC0555-9187-4F99-A721-F5228F14BCFCQ52659149-3F71CE48-A83E-42F2-8C5A-1419D0740D5DQ55646811-7E1C24F2-D78F-4D40-814C-E47D42FD2105Q58099592-A7269979-B875-453E-8BDC-5B8AB8AB24A2Q58798205-60F4CEAF-4578-4329-9522-A8DE1CC8B7E4Q59138260-46F17683-9861-43DC-B256-00CDF9090FFE
P2860
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
description
2015 nî lūn-bûn
@nan
2015年の論文
@ja
2015年学术文章
@wuu
2015年学术文章
@zh-cn
2015年学术文章
@zh-hans
2015年学术文章
@zh-my
2015年学术文章
@zh-sg
2015年學術文章
@yue
2015年學術文章
@zh
2015年學術文章
@zh-hant
name
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
@ast
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
@en
type
label
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
@ast
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
@en
prefLabel
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
@ast
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
@en
P2093
P2860
P356
P1476
Agonism, Antagonism, and Inverse Agonism Bias at the Ghrelin Receptor Signaling
@en
P2093
Aude Saulière
Céline Galés
Céline M'Kadmi
Didier Gagne
Jacky Marie
Jean-Alain Fehrentz
Jean-Louis Banères
Jean-Philippe Leyris
Lauriane Onfroy
Marjorie Damian
P2860
P304
27021-27039
P356
10.1074/JBC.M115.659250
P407
P577
2015-09-11T00:00:00Z