Pharmacological blockade of the cold receptor TRPM8 attenuates autonomic and behavioral cold defenses and decreases deep body temperature.
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Antibodies to the extracellular pore loop of TRPM8 act as antagonists of channel activationHibernation, Hypothermia and a Possible Therapeutic "Shifted Homeostasis" Induced by Central Activation of A1 Adenosine Receptor (A1AR)Central control of body temperatureInduction of therapeutic hypothermia by pharmacological modulation of temperature-sensitive TRP channels: theoretical framework and practical considerationsSpecies-specific temperature sensitivity of TRPA1TRPM3 in temperature sensing and beyondTRP ion channels in thermosensation, thermoregulation and metabolismVAMP7 regulates constitutive membrane incorporation of the cold-activated channel TRPM8.Spinal cord thermosensitivity: An afferent phenomenon?Molecular mechanisms of temperature adaptationExpression of temperature-sensitive ion channel TRPM8 in sperm cells correlates with vertebrate evolutionNeural Signaling Metabolites May Modulate Energy Use in Hibernation.Skin temperature: its role in thermoregulationIn vivo correlates of thermoregulatory defense in humans: Temporal course of sub-cortical and cortical responses assessed with fMRI.Development of TRPM8 Antagonists to Treat Chronic Pain and Migraine.Local daily temperatures, thermal seasons, and suicide rates in Finland from 1974 to 2010.Cold-Induced Thermogenesis and Inflammation-Associated Cold-Seeking Behavior Are Represented by Different Dorsomedial Hypothalamic Sites: A Three-Dimensional Functional Topography Study in Conscious RatsThe TRPM8 protein is a testosterone receptor: II. Functional evidence for an ionotropic effect of testosterone on TRPM8AMG2850, a potent and selective TRPM8 antagonist, is not effective in rat models of inflammatory mechanical hypersensitivity and neuropathic tactile allodyniaTRPM8 on mucosal sensory nerves regulates colitogenic responses by innate immune cells via CGRPCentral nervous system regulation of brown adipose tissue.Meningeal transient receptor potential channel M8 activation causes cutaneous facial and hindpaw allodynia in a preclinical rodent model of headacheCurrent understanding on the neurophysiology of behavioral thermoregulation."Science without Borders" program and Brazilian-Hungarian collaboration in thermoregulation.Brazil: What country is this?The role of trigeminal nasal TRPM8-expressing afferent neurons in the antitussive effects of menthol.An animal model of oxaliplatin-induced cold allodynia reveals a crucial role for Nav1.6 in peripheral pain pathwaysLipopolysaccharide-induced neuronal activation in the paraventricular and dorsomedial hypothalamus depends on ambient temperature.Shivering and tachycardic responses to external cooling in mice are substantially suppressed by TRPV1 activation but not by TRPM8 inhibition.Autonomic regulation of brown adipose tissue thermogenesis in health and disease: potential clinical applications for altering BAT thermogenesis.Transient receptor potential channel ankyrin-1 is not a cold sensor for autonomic thermoregulation in rodents.TRPM8 and MigraineCentral actions of somatostatin-28 and oligosomatostatin agonists to prevent components of the endocrine, autonomic and visceral responses to stress through interaction with different somatostatin receptor subtypes.Genes, molecules and patients--emerging topics to guide clinical pain research.TRPV1, TRPA1, and TRPM8 channels in inflammation, energy redirection, and water retention: role in chronic inflammatory diseases with an evolutionary perspective.Transient receptor potential channel modulators as pharmacological treatments for lower urinary tract symptoms (LUTS): myth or reality?A vascular mechanistic approach to understanding Raynaud phenomenon.Emerging drugs for overactive bladder.Body Temperature Measurements for Metabolic Phenotyping in Mice.Involvement of thermosensitive TRP channels in energy metabolism.
P2860
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P2860
Pharmacological blockade of the cold receptor TRPM8 attenuates autonomic and behavioral cold defenses and decreases deep body temperature.
description
2012 nî lūn-bûn
@nan
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
2012年论文
@zh
2012年论文
@zh-cn
name
Pharmacological blockade of th ...... creases deep body temperature.
@ast
Pharmacological blockade of th ...... creases deep body temperature.
@en
type
label
Pharmacological blockade of th ...... creases deep body temperature.
@ast
Pharmacological blockade of th ...... creases deep body temperature.
@en
prefLabel
Pharmacological blockade of th ...... creases deep body temperature.
@ast
Pharmacological blockade of th ...... creases deep body temperature.
@en
P2093
P2860
P1476
Pharmacological blockade of th ...... creases deep body temperature.
@en
P2093
Andrej A Romanovsky
Daniela L Oliveira
Diana Bautista
M Camila Almeida
Narender R Gavva
Nuria Tamayo
Prafulla Aryal
Renato N Soriano
P2860
P304
P356
10.1523/JNEUROSCI.5606-11.2012
P407
P577
2012-02-01T00:00:00Z