Thiophene-core estrogen receptor ligands having superagonist activity. - sprookjes - yvandenbroek - TriplyDB

Thiophene-core estrogen receptor ligands having superagonist activity.

Thiophene-core estrogen receptor ligands having superagonist activity.

http://www.wikidata.org/entity/Q36883747

about

Selenophene and thiophene-core estrogen receptor ligands that inhibit motility and development of parasitic stages of Haemonchus contortus.Predictive features of ligand-specific signaling through the estrogen receptor Synthesis and receptor binding in trans-CD ring-fused A-CD estrogens: comparison with the cis-fused isomers.Selective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast Cancer Triaryl-substituted Schiff bases are high-affinity subtype-selective ligands for the estrogen receptor.Site-selective Suzuki-Miyaura coupling of heteroaryl halides - understanding the trends for pharmaceutically important classes.Selenophenes: Introducing a New Element into the Core of Non-Steroidal Estrogen Receptor Ligands.Novel synthesis of 5-methyl-5,10-dihydroindolo[3,2-b]indoles by Pd-catalyzed C-C and two-fold C-N coupling reactions.Water compatible multicomponent cascade Suzuki/Heck-aldol, Suzuki-aldol-Suzuki, and aldol-Suzuki-aldol reactions: an ecofriendly paradigm for multiple carbon-carbon bond formation in one pot.

P2860

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P2860

Thiophene-core estrogen receptor ligands having superagonist activity.

http://www.wikidata.org/entity/Q36883747

description

2013 nî lūn-bûn

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2013年の論文

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2013年論文

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2013年論文

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2013年論文

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2013年論文

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2013年論文

@zh-tw

2013年论文

@wuu

2013年论文

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2013年论文

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name

Thiophene-core estrogen receptor ligands having superagonist activity.

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type

label

Thiophene-core estrogen receptor ligands having superagonist activity.

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prefLabel

Thiophene-core estrogen receptor ligands having superagonist activity.

@en

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P1433

Journal of Medicinal Chemistry

P1476

Thiophene-core estrogen receptor ligands having superagonist activity

@en

P2093

Jian Min

http://www.w3.org/2001/XMLSchema#string

John A Katzenellenbogen

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Kathryn E Carlson

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Kendall W Nettles

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Minjian Huang

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Sathish Srinivasan

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P2860

Cloning of a novel receptor expressed in rat prostate and ovary

Resveratrol, a polyphenolic compound found in grapes and wine, is an agonist for the estrogen receptor

Estrogen receptors and human disease

Estrogen Receptors alpha and beta as determinants of gene expression: influence of ligand, dose, and chromatin binding

Estrogen receptor transcription and transactivation: Estrogen receptor alpha and estrogen receptor beta: regulation by selective estrogen receptor modulators and importance in breast cancer.

Structure of the ligand-binding domain of oestrogen receptor beta in the presence of a partial agonist and a full antagonist

Development of Selective Estrogen Receptor Modulator (SERM)-Like Activity Through an Indirect Mechanism of Estrogen Receptor Antagonism: Defining the Binding Mode of 7-Oxabicyclo[2.2.1]hept-5-ene Scaffold Core Ligands

Molecular basis of agonism and antagonism in the oestrogen receptor

Coot: model-building tools for molecular graphics

Synthesis and pharmacological evaluation of 1H-imidazoles as ligands for the estrogen receptor and cytotoxic inhibitors of the cyclooxygenase

P304

3346-3366

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scholarly article

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10.1021/JM400157E

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8

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56

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Jerome C Nwachukwu

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2013-04-15T00:00:00Z

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