The prevalence, maintenance, and relevance of G protein-coupled receptor oligomerization
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Membrane omega-3 fatty acids modulate the oligomerisation kinetics of adenosine A2A and dopamine D2 receptors.A G Protein-Coupled Receptor Dimerization Interface in Human Cone OpsinsFluorescence correlation spectroscopy analysis of serotonin, adrenergic, muscarinic, and dopamine receptor dimerization: the oligomer number puzzleTime-resolved fluorescence spectroscopy measures clustering and mobility of a G protein-coupled receptor opsin in live cell membranesCoupling of g proteins to reconstituted monomers and tetramers of the M2 muscarinic receptorCB2 Cannabinoid receptors as a therapeutic target-what does the future hold?Functional selectivity of allosteric interactions within G protein-coupled receptor oligomers: the dopamine D1-D3 receptor heterotetramer.Opportunities and challenges in the discovery of allosteric modulators of GPCRs for treating CNS disorders.Dynamic Regulation of Quaternary Organization of the M1 Muscarinic Receptor by Subtype-selective Antagonist Drugs.Descending control of itch transmission by the serotonergic system via 5-HT1A-facilitated GRP-GRPR signalingStoichiometry and geometry of the CXC chemokine receptor 4 complex with CXC ligand 12: molecular modeling and experimental validation.Native serotonin 5-HT2C receptors are expressed as homodimers on the apical surface of choroid plexus epithelial cellsImproved methodical approach for quantitative BRET analysis of G Protein Coupled Receptor dimerizationPhage display and hybridoma generation of antibodies to human CXCR2 yields antibodies with distinct mechanisms and epitopes.Regulation of oligomeric organization of the serotonin 5-hydroxytryptamine 2C (5-HT2C) receptor observed by spatial intensity distribution analysisDistinct Agonist Regulation of Muscarinic Acetylcholine M2-M3 Heteromers and Their Corresponding Homomers.Taking two to tango: a role for ghrelin receptor heterodimerization in stress and reward.Novel structural and functional insights into M3 muscarinic receptor dimer/oligomer formation.G protein-coupled receptor oligomerization revisited: functional and pharmacological perspectives.EuroTracker® dyes: design, synthesis, structure and photophysical properties of very bright europium complexes and their use in bioassays and cellular optical imaging.Revealing G-protein-coupled receptor oligomerization at the single-molecule level through a nanoscopic lens: methods, dynamics and biological function.Allosteric Modulation of GPCRs: New Insights and Potential Utility for Treatment of Schizophrenia and Other CNS Disorders.Breaking barriers to novel analgesic drug development.Hallucinogens and Serotonin 5-HT2A Receptor-Mediated Signaling Pathways.HSV-Mediated Transgene Expression of Chimeric Constructs to Study Behavioral Function of GPCR Heteromers in Mice.Analysis of Human Dopamine D3 Receptor Quaternary Structure.Structure and Function of Cross-class Complexes of G Protein-coupled Secretin and Angiotensin 1a Receptors.Nanoscale high-content analysis using compositional heterogeneities of single proteoliposomes.Spatial intensity distribution analysis quantifies the extent and regulation of homodimerization of the secretin receptor.A Molecular Basis for Selective Antagonist Destabilization of Dopamine D3 Receptor Quaternary Organization.Quaternary structures of opsin in live cells revealed by FRET spectrometry.Family a GPCR heteromers in animal models.[G protein-coupled receptors in the spot light].Muscarinic receptor oligomerization.P2Y11 Receptors: Properties, Distribution and Functions.Using Biosensors to Study Free Fatty Acid Receptor Pharmacology and Function.Bright, Highly Water-Soluble Triazacyclononane Europium Complexes To Detect Ligand Binding with Time-Resolved FRET MicroscopyBright, Highly Water-Soluble Triazacyclononane Europium Complexes To Detect Ligand Binding with Time-Resolved FRET Microscopy
P2860
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P2860
The prevalence, maintenance, and relevance of G protein-coupled receptor oligomerization
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
2013年论文
@zh
2013年论文
@zh-cn
name
The prevalence, maintenance, and relevance of G protein-coupled receptor oligomerization
@en
type
label
The prevalence, maintenance, and relevance of G protein-coupled receptor oligomerization
@en
prefLabel
The prevalence, maintenance, and relevance of G protein-coupled receptor oligomerization
@en
P2860
P356
P1476
The prevalence, maintenance, and relevance of G protein-coupled receptor oligomerization
@en
P2093
Graeme Milligan
P2860
P304
P356
10.1124/MOL.113.084780
P577
2013-04-30T00:00:00Z