Dihydropyrimidinone positive modulation of delta-subunit-containing gamma-aminobutyric acid type A receptors, including an epilepsy-linked mutant variant.
about
A study of subunit selectivity, mechanism and site of action of the delta selective compound 2 (DS2) at human recombinant and rodent native GABA(A) receptors.Etomidate produces similar allosteric modulation in α1β3δ and α1β3γ2L GABA(A) receptors.Use of multicomponent reactions in developing small-molecule tools to study GABAA receptor mechanism and function.Allosteric Modulation of αβδ GABAA Receptors.
P2860
Dihydropyrimidinone positive modulation of delta-subunit-containing gamma-aminobutyric acid type A receptors, including an epilepsy-linked mutant variant.
description
article científic
@ca
article scientifique
@fr
articolo scientifico
@it
artigo científico
@pt
bilimsel makale
@tr
scientific article published on June 2010
@en
vedecký článok
@sk
vetenskaplig artikel
@sv
videnskabelig artikel
@da
vědecký článek
@cs
name
Dihydropyrimidinone positive m ...... pilepsy-linked mutant variant.
@en
Dihydropyrimidinone positive m ...... pilepsy-linked mutant variant.
@nl
type
label
Dihydropyrimidinone positive m ...... pilepsy-linked mutant variant.
@en
Dihydropyrimidinone positive m ...... pilepsy-linked mutant variant.
@nl
prefLabel
Dihydropyrimidinone positive m ...... pilepsy-linked mutant variant.
@en
Dihydropyrimidinone positive m ...... pilepsy-linked mutant variant.
@nl
P2093
P2860
P356
P1433
P1476
Dihydropyrimidinone positive m ...... pilepsy-linked mutant variant.
@en
P2093
Bruce Ganem
George P Hess
Jason G Polisar
John Mabry
Kyle P Eagen
Ryan W Lewis
P2860
P304
P356
10.1021/BI100119T
P407
P577
2010-06-01T00:00:00Z