Linsitinib (OSI-906) antagonizes ATP-binding cassette subfamily G member 2 and subfamily C member 10-mediated drug resistance.
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Repositioning of Tyrosine Kinase Inhibitors as Antagonists of ATP-Binding Cassette Transporters in Anticancer Drug ResistanceSynthesis and biological evaluation of pentacyclic strychnos alkaloids as selective modulators of the ABCC10 (MRP7) efflux pumpWHI-P154 enhances the chemotherapeutic effect of anticancer agents in ABCG2-overexpressing cells.The small molecule tyrosine kinase inhibitor NVP-BHG712 antagonizes ABCC10-mediated paclitaxel resistance: a preclinical and pharmacokinetic study.A-803467, a tetrodotoxin-resistant sodium channel blocker, modulates ABCG2-mediated MDR in vitro and in vivo.Thiazole-valine peptidomimetic (TTT-28) antagonizes multidrug resistance in vitro and in vivo by selectively inhibiting the efflux activity of ABCB1.Tyrosine kinase inhibitors as reversal agents for ABC transporter mediated drug resistance.Modulating the function of ATP-binding cassette subfamily G member 2 (ABCG2) with inhibitor cabozantinib.ABCG2/BCRP: Specific and Nonspecific Modulators.Tyrosine kinase inhibitors enhanced the efficacy of conventional chemotherapeutic agent in multidrug resistant cancer cells.Regorafenib overcomes chemotherapeutic multidrug resistance mediated by ABCB1 transporter in colorectal cancer: In vitro and in vivo study.2-Trifluoromethyl-2-Hydroxypropionamide Derivatives as Novel Reversal Agents of ABCG2 (BCRP)-Mediated Multidrug Resistance: Synthesis and Biological Evaluations.
P2860
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P2860
Linsitinib (OSI-906) antagonizes ATP-binding cassette subfamily G member 2 and subfamily C member 10-mediated drug resistance.
description
2014 nî lūn-bûn
@nan
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
2014年论文
@zh
2014年论文
@zh-cn
name
Linsitinib (OSI-906) antagoniz ...... r 10-mediated drug resistance.
@en
Linsitinib
@nl
type
label
Linsitinib (OSI-906) antagoniz ...... r 10-mediated drug resistance.
@en
Linsitinib
@nl
prefLabel
Linsitinib (OSI-906) antagoniz ...... r 10-mediated drug resistance.
@en
Linsitinib
@nl
P2093
P1476
Linsitinib (OSI-906) antagoniz ...... er 10-mediated drug resistance
@en
P2093
Charles R Ashby
Rishil J Kathawala
Suneet Shukla
Suresh V Ambudkar
Susan E Bates
Tanaji T Talele
Yi-Jun Wang
Yun-Kai Zhang
P304
P356
10.1016/J.BIOCEL.2014.03.026
P577
2014-04-12T00:00:00Z