Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal?
about
The Dipeptidyl Peptidase Family, Prolyl Oligopeptidase, and Prolyl Carboxypeptidase in the Immune System and Inflammatory Disease, Including AtherosclerosisAn essential signal peptide peptidase identified in an RNAi screen of serine peptidases of Trypanosoma bruceiEfficient access to enantiopure 1,3-disubstituted isoindolines from selective catalytic fragmentation of an original desymmetrized rigid overbred templateGrassypeptolides as natural inhibitors of dipeptidyl peptidase 8 and T-cell activation.Targeted inactivation of dipeptidyl peptidase 9 enzymatic activity causes mouse neonate lethality.Regulation of dipeptidyl peptidase 8 and 9 expression in activated lymphocytes and injured liver.Novel hydrazine derivatives as selective DPP-IV inhibitors: findings from virtual screening and validation through molecular dynamics simulations.The Dipeptidyl Peptidases 4, 8, and 9 in Mouse Monocytes and Macrophages: DPP8/9 Inhibition Attenuates M1 Macrophage Activation in Mice.Selective Inhibitors of Fibroblast Activation Protein (FAP) with a (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine Scaffold.DPP9 is a novel component of the N-end rule pathway targeting the tyrosine kinase Syk.The SUMO1-E67 interacting loop peptide is an allosteric inhibitor of the dipeptidyl peptidases 8 and 9.A novel SUMO1-specific interacting motif in dipeptidyl peptidase 9 (DPP9) that is important for enzymatic regulation.Dipeptidyl peptidases in atherosclerosis: expression and role in macrophage differentiation, activation and apoptosis.Fibroblast activation protein-α in fibrogenic disorders and cancer: more than a prolyl-specific peptidase?Structures and mechanism of dipeptidyl peptidases 8 and 9, important players in cellular homeostasis and cancer.Probing for improved selectivity with dipeptide-derived inhibitors of dipeptidyl peptidases 8 and 9: the impact of P1-variationSelective inhibitors of fibroblast activation protein (FAP) with a xanthine scaffoldSynthesis of γ,δ-Aziridino α-Amino Acid Derivatives and their Stereoselective Ring Transformation to 2-(Aminomethyl)-1-aminocyclopropanecarboxylic Acid Derivatives
P2860
Q26795473-AF7A7976-DCC6-47FF-8763-1E4168EC4763Q28545105-1A8FD119-D6A3-435C-88A3-47441247FB3AQ29031161-132E398B-BC10-48E6-A626-BEE112CCBBECQ33728657-996E42EC-725D-41B5-9000-9A40D9F454C7Q35040181-6F0D6082-A20E-4654-BABF-A282A53B61C4Q36865097-43FFE239-AE07-4503-AC5C-D28D84B289C5Q38398676-6694E649-B8ED-4253-A2E3-B8DB513E5AAEQ38828981-76010110-2CDA-4934-B0D4-960F3CE8A034Q39769132-B8007F63-8AFF-44E4-A1FE-0FB4EEF77871Q41199050-086ACFE0-78A0-47DF-B3A0-24DDBD973660Q42134616-7A6C065A-AC3E-4520-B8A1-3AC8637DE358Q42269173-FC87D4D1-BF75-4D25-9159-5E2E69FB5AF4Q45897317-BEB9F431-1C04-4D84-91A1-79D318E03E06Q47922336-593AA8D5-59DE-43E2-B91C-CF9F78ADA1CDQ48139349-7E607FF2-2410-4B0A-AA46-13DCD722E19DQ58864159-88685132-9518-4798-893D-BB34C38416E7Q58864169-02678A69-6A67-4D4C-BE19-F63FA3CA3964Q58864171-AE2744B1-74B8-4650-87B8-9A05C2F2768F
P2860
Structure-activity relationship studies on isoindoline inhibitors of dipeptidyl peptidases 8 and 9 (DPP8, DPP9): is DPP8-selectivity an attainable goal?
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年学术文章
@wuu
2011年学术文章
@zh-cn
2011年学术文章
@zh-hans
2011年学术文章
@zh-my
2011年学术文章
@zh-sg
2011年學術文章
@yue
2011年學術文章
@zh
2011年學術文章
@zh-hant
name
Structure-activity relationshi ...... electivity an attainable goal?
@en
Structure-activity relationshi ...... electivity an attainable goal?
@nl
type
label
Structure-activity relationshi ...... electivity an attainable goal?
@en
Structure-activity relationshi ...... electivity an attainable goal?
@nl
prefLabel
Structure-activity relationshi ...... electivity an attainable goal?
@en
Structure-activity relationshi ...... electivity an attainable goal?
@nl
P2093
P50
P356
P1476
Structure-activity relationshi ...... electivity an attainable goal?
@en
P2093
Achiel Haemers
Jurgen Joossens
Sebastiaan Van Goethem
Veerle Matheeussen
P304
P356
10.1021/JM200383J
P407
P577
2011-08-02T00:00:00Z