Facilitation of μ-opioid receptor activity by preventing δ-opioid receptor-mediated codegradation.
about
The δ opioid receptor agonist SNC80 selectively activates heteromeric μ-δ opioid receptorsOpioid receptor trafficking and interaction in nociceptorsAntibodies to probe endogenous G protein-coupled receptor heteromer expression, regulation, and functionOpioid receptors: toward separation of analgesic from undesirable effectsOpioid receptor heteromers in analgesiaThe functional and anatomical dissection of somatosensory subpopulations using mouse geneticsPreferred supramolecular organization and dimer interfaces of opioid receptors from simulated self-associationCrystal structure of the µ-opioid receptor bound to a morphinan antagonistAllosteric mechanisms within the adenosine A2A-dopamine D2 receptor heterotetramerCircadian-related heteromerization of adrenergic and dopamine D₄ receptors modulates melatonin synthesis and release in the pineal glandAnti-analgesic effect of the mu/delta opioid receptor heteromer revealed by ligand-biased antagonismBerberine Improves Intestinal Motility and Visceral Pain in the Mouse Models Mimicking Diarrhea-Predominant Irritable Bowel Syndrome (IBS-D) Symptoms in an Opioid-Receptor Dependent MannerDelta opioid receptors presynaptically regulate cutaneous mechanosensory neuron input to the spinal cord dorsal horn.Emergence of functional spinal delta opioid receptors after chronic ethanol exposureContribution of mu and delta opioid receptors to the pharmacological profile of kappa opioid receptor subtypes.A heroin addiction severity-associated intronic single nucleotide polymorphism modulates alternative pre-mRNA splicing of the μ opioid receptor gene OPRM1 via hnRNPH interactions.Functional selectivity of allosteric interactions within G protein-coupled receptor oligomers: the dopamine D1-D3 receptor heterotetramer.Identification of a μ-δ opioid receptor heteromer-biased agonist with antinociceptive activity.Revolution in GPCR signalling: opioid receptor heteromers as novel therapeutic targets: IUPHAR review 10.Novel screening assay for the selective detection of G-protein-coupled receptor heteromer signaling.Mix and match: heterodimers and opioid tolerance.Dimerization with cannabinoid receptors allosterically modulates delta opioid receptor activity during neuropathic pain.Differential response to morphine of the oligomeric state of μ-opioid in the presence of δ-opioid receptorsHeteromers of μ-δ opioid receptors: new pharmacology and novel therapeutic possibilities.Analgesic synergy between opioid and α2 -adrenoceptorsRecent advances on the δ opioid receptor: from trafficking to function.In vivo opioid receptor heteromerization: where do we stand?Prolonged morphine treatment alters δ opioid receptor post-internalization traffickingLigand requirements for involvement of PKCε in synergistic analgesic interactions between spinal μ and δ opioid receptors.GPCR Heterodimerization in the Reproductive System: Functional Regulation and Implication for BiodiversityHeteromerization of the μ- and δ-opioid receptors produces ligand-biased antagonism and alters μ-receptor traffickingDifferential stability of the crystallographic interfaces of mu- and kappa-opioid receptorsMuscarinic acetylcholine receptor M3 modulates odorant receptor activity via inhibition of β-arrestin-2 recruitment.Implication of delta opioid receptor subtype 2 but not delta opioid receptor subtype 1 in the development of morphine analgesic tolerance in a rat model of chronic inflammatory pain.Orexin-corticotropin-releasing factor receptor heteromers in the ventral tegmental area as targets for cocaineEngineering endomorphin drugs: state of the art.Characterisation of the Novel Mixed Mu-NOP Peptide Ligand Dermorphin-N/OFQ (DeNo).Opioid receptors: Structural and mechanistic insights into pharmacology and signaling.Ubiquitination of G protein-coupled receptors: functional implications and drug discovery.Minireview: ubiquitination-regulated G protein-coupled receptor signaling and trafficking
P2860
Q24630886-E69E0E94-EB6D-4A4D-B065-B079E733E964Q26822251-FCB039E2-0941-4048-A7A8-12661E690BB5Q26992192-8DF2C9E7-1AF3-4079-8A42-C1DF28F78C21Q27002925-D8BC8D56-A789-4902-9984-6A33663A339FQ27004306-B1FE0590-623C-4B28-B666-89569C5F9905Q27014891-4970A386-1760-4243-820B-6BC4E09C48FBQ27319797-2570D4A6-36FC-4964-A458-05874D4893D0Q27678133-46C7E9D3-5E54-4273-B2DA-AE65EB1696D2Q28263053-6D346653-0667-41BE-A30F-FE2C2FD177D1Q28480542-ED04EA43-E13C-44FE-BFAB-64D50829A26EQ28488120-6889AF5F-0952-4BB7-80EF-344E19C8EA82Q28551749-20F8A5D8-E310-4516-9DD0-D5559C236C78Q33811673-BE4094B0-BBAE-4DEB-8AB1-2964A381C492Q33863121-FA29EC61-E93A-4D3B-8991-DFA44064B742Q33863139-A0A7ACC1-9C98-4655-8C74-7F2CE1F986CEQ34037595-6C83204B-D63A-42AD-BDC2-9E83ED556EFBQ34186022-006B4970-4CC2-4D03-98BA-960581C9AFB0Q34354902-17596E49-C790-4175-AABC-AA6B45151BE6Q34424009-CEF99F83-D7A4-42D1-BB29-B9925BA632E1Q34457615-0ED46C04-11A9-43B3-BCBC-6B79636B9452Q34522291-CAC107F4-7925-4067-A1E3-854E085ADAFFQ34524896-4E9F056A-AB0C-4A9C-9CC2-1F8439A3E8EAQ34767171-DE2C3EA0-640A-490D-BDEF-2DF1BDD3D967Q34939624-72266AB4-AE82-48B0-A91F-DCE4D3545285Q34939644-6B0732FD-F2F9-4DF6-A217-29DD0D50E09BQ34939664-1434FF0C-A5F6-4933-811D-E6C885C9CD16Q34939677-44FD7C19-2CD2-42B4-97CC-57839F0034A1Q34939888-775B9CEC-D852-41E2-856A-A3218E657BEBQ34939914-5717E2E9-D867-4E97-92C9-5B5DE94BA0C9Q34962059-826FFFFF-9065-48DB-BBA7-ADAA8A6ADDF2Q34989880-A9FA99B4-358D-44E6-8353-326BF567B8A0Q35126350-222F8588-A359-4634-A0EE-E915458F2E9FQ35214958-C9FCAFAC-26C8-4090-BFA6-35A7EC347906Q35327954-F7C9A333-063C-40A2-AE08-12158B738EC3Q35547856-3FD83DE8-CA10-4ACF-8E22-557F4F02A66AQ35660653-3AAFC347-2BBF-4E58-A59C-0235F2FAC79BQ36043728-1DE13AA0-E0CA-4F7D-AE7B-3EBF28B5A6E3Q36096058-016AEED8-E2F0-4E00-9BBF-C64F9A3ECE04Q36294416-5CC105D4-E043-41B1-A5A2-881BE692DBF7Q36714881-A047B164-13D7-49B2-A945-A7ADB8CDFD91
P2860
Facilitation of μ-opioid receptor activity by preventing δ-opioid receptor-mediated codegradation.
description
2011 nî lūn-bûn
@nan
2011年の論文
@ja
2011年学术文章
@wuu
2011年学术文章
@zh
2011年学术文章
@zh-cn
2011年学术文章
@zh-hans
2011年学术文章
@zh-my
2011年学术文章
@zh-sg
2011年學術文章
@yue
2011年學術文章
@zh-hant
name
Facilitation of μ-opioid recep ...... ceptor-mediated codegradation.
@en
Facilitation of μ-opioid recep ...... ceptor-mediated codegradation.
@nl
type
label
Facilitation of μ-opioid recep ...... ceptor-mediated codegradation.
@en
Facilitation of μ-opioid recep ...... ceptor-mediated codegradation.
@nl
prefLabel
Facilitation of μ-opioid recep ...... ceptor-mediated codegradation.
@en
Facilitation of μ-opioid recep ...... ceptor-mediated codegradation.
@nl
P2093
P1433
P1476
Facilitation of μ-opioid recep ...... eceptor-mediated codegradation
@en
P2093
Hai-Bo Wang
Hong-Rui Liu
Qiong Wang
Shao-Qiu He
Ying-Jin Lu
P304
P356
10.1016/J.NEURON.2010.12.001
P407
P577
2011-01-01T00:00:00Z