A Novel Negative Allosteric Modulator Selective for GluN2C/2D-Containing NMDA Receptors Inhibits Synaptic Transmission in Hippocampal Interneurons.
about
The bioactive protein-ligand conformation of GluN2C-selective positive allosteric modulators bound to the NMDA receptor.NMDA receptor blockade ameliorates abnormalities of spike firing of subthalamic nucleus neurons in a parkinsonian nonhuman primate.An NMDAR positive and negative allosteric modulator series share a binding site and are interconverted by methyl groups.Higher ambient synaptic glutamate at inhibitory versus excitatory neurons differentially impacts NMDA receptor activityA structurally derived model of subunit-dependent NMDA receptor function
P2860
A Novel Negative Allosteric Modulator Selective for GluN2C/2D-Containing NMDA Receptors Inhibits Synaptic Transmission in Hippocampal Interneurons.
description
2017 nî lūn-bûn
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2017年の論文
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2017年学术文章
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2017年学术文章
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2017年学术文章
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2017年学术文章
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name
A Novel Negative Allosteric Mo ...... n in Hippocampal Interneurons.
@en
A Novel Negative Allosteric Mo ...... n in Hippocampal Interneurons.
@nl
type
label
A Novel Negative Allosteric Mo ...... n in Hippocampal Interneurons.
@en
A Novel Negative Allosteric Mo ...... n in Hippocampal Interneurons.
@nl
prefLabel
A Novel Negative Allosteric Mo ...... n in Hippocampal Interneurons.
@en
A Novel Negative Allosteric Mo ...... n in Hippocampal Interneurons.
@nl
P2093
P2860
P50
P1476
A Novel Negative Allosteric Mo ...... on in Hippocampal Interneurons
@en
P2093
Cara A Mosley
Christoffer Bundgaard
David S Menaldino
Henrik S Jensen
John O DiRaddo
Katie M Vance
Samantha L Summer
Scott J Myers
Sommer S Zimmerman
Timothy M Acker
P2860
P304
P356
10.1021/ACSCHEMNEURO.7B00329
P577
2017-11-02T00:00:00Z