HU-243
HU-243 (AM-4056) is a synthetic cannabinoid drug that is a single enantiomer of the hydrogenated derivative of the commonly used reference agonist HU-210. It is a methylene homologue of canbisol. It is a potent agonist at both the CB1 and CB2 receptors, with a binding affinity of 0.041 nM at the CB1 receptor, making it marginally more potent than HU-210, which had an affinity of 0.061 nM in the same assay.
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HU-243
HU-243 (AM-4056) is a synthetic cannabinoid drug that is a single enantiomer of the hydrogenated derivative of the commonly used reference agonist HU-210. It is a methylene homologue of canbisol. It is a potent agonist at both the CB1 and CB2 receptors, with a binding affinity of 0.041 nM at the CB1 receptor, making it marginally more potent than HU-210, which had an affinity of 0.061 nM in the same assay.
has abstract
HU-243 (AM-4056) is a syntheti ...... of 0.061 nM in the same assay.
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CAS number
140835-18-3
PubChem
Wikipage page ID
28,806,935
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1,022,958,079
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CAS number
IUPAC name
IUPHAR ligand
PubChem
SMILES
CC[C@H]2[C@@H]C3=C1C=CC=C3O
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hypernym
comment
HU-243 (AM-4056) is a syntheti ...... of 0.061 nM in the same assay.
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label
HU-243
@en