Flexible modulation of agonist efficacy at the human A3 adenosine receptor by the imidazoquinoline allosteric enhancer LUF6000
about
UDP-glucose acting at P2Y14 receptors is a mediator of mast cell degranulationA₃ adenosine receptor allosteric modulator induces an anti-inflammatory effect: in vivo studies and molecular mechanism of action.Modulation of A1 and A2B adenosine receptor activity: a new strategy to sensitise glioblastoma stem cells to chemotherapy.International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and classification of adenosine receptors--an updateFunctionally biased modulation of A(3) adenosine receptor agonist efficacy and potency by imidazoquinolinamine allosteric enhancersAllosteric modulation of purine and pyrimidine receptors.Protection from myocardial ischemia/reperfusion injury by a positive allosteric modulator of the A₃ adenosine receptor.Introduction to adenosine receptors as therapeutic targets.Functional selectivity of adenosine A1 receptor ligands?Allosteric modulation and functional selectivity of G protein-coupled receptors.Soluble ecto-5'-nucleotidase (5'-NT), alkaline phosphatase, and adenosine deaminase (ADA1) activities in neonatal blood favor elevated extracellular adenosine.Novel 2- and 4-substituted 1H-imidazo[4,5-c]quinolin-4-amine derivatives as allosteric modulators of the A3 adenosine receptorAllosteric ligands for G protein-coupled receptors: a novel strategy with attractive therapeutic opportunities.Progress towards novel adenosine receptor therapeutics gleaned from the recent patent literature.The A3 adenosine receptor as multifaceted therapeutic target: pharmacology, medicinal chemistry, and in silico approaches.A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.Species differences and mechanism of action of A3 adenosine receptor allosteric modulators.Prediction of consensus binding mode geometries for related chemical series of positive allosteric modulators of adenosine and muscarinic acetylcholine receptors.
P2860
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P2860
Flexible modulation of agonist efficacy at the human A3 adenosine receptor by the imidazoquinoline allosteric enhancer LUF6000
description
2008 nî lūn-bûn
@nan
2008 թուականին հրատարակուած գիտական յօդուած
@hyw
2008 թվականին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@ast
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@en
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@en-gb
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@nl
type
label
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@ast
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@en
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@en-gb
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@nl
prefLabel
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@ast
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@en
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@en-gb
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@nl
P2860
P50
P356
P1433
P1476
Flexible modulation of agonist ...... ne allosteric enhancer LUF6000
@en
P2093
P2860
P2888
P356
10.1186/1471-2210-8-20
P407
P577
2008-01-01T00:00:00Z
P5875
P6179
1032549338