SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats - Wikidata - awgldk - TriplyDB

SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

http://www.wikidata.org/entity/Q24672651

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Serotonin 5-HT7 receptor agents: Structure-activity relationships and potential therapeutic applications in central nervous system disorders Amisulpride is a potent 5-HT7 antagonist: relevance for antidepressant actions in vivo The role of the serotonin receptor subtypes 5-HT1A and 5-HT7 and its interaction in emotional learning and memory Review of pharmacological treatment in mood disorders and future directions for drug development.Genome-wide association discoveries of alcohol dependence Targeting the Serotonin 5-HT7 Receptor in the Search for Treatments for CNS Disorders: Rationale and Progress to Date Dual- and triple-acting agents for treating core and co-morbid symptoms of major depression: novel concepts, new drugs Evidence for the involvement of central 5-HT7 receptors in the micturition reflex in anaesthetized female rats Pharmacological blockade of 5-HT7 receptors as a putative fast acting antidepressant strategy Molecular targets for treating cognitive dysfunction in schizophrenia.Inactivation of the 5-HT(7) receptor partially blocks phencyclidine-induced disruption of prepulse inhibition.The 5-HT7 receptor and disorders of the nervous system: an overview.5-HT7 receptors as modulators of neuronal excitability, synaptic transmission and plasticity: physiological role and possible implications in autism spectrum disorders.Role of the 5-HT7 receptor in the central nervous system: from current status to future perspectives.Interplay between serotonin 5-HT1A and 5-HT7 receptors in depressive disorders.Differentiated effects of the multimodal antidepressant vortioxetine on sleep architecture: Part 2, pharmacological interactions in rodents suggest a role of serotonin-3 receptor antagonism.Autoradiographic distribution of 5-HT7 receptors in the human brain using [3H]mesulergine: comparison to other mammalian species.Genome-wide association study of theta band event-related oscillations identifies serotonin receptor gene HTR7 influencing risk of alcohol dependence.Expression of 5-HT7 receptor mRNA in the hamster brain: effect of aging and association with calbindin-D28K expression.Vagal control of the heart: central serotonergic (5-HT) mechanisms.5-HT7R/G12 signaling regulates neuronal morphology and function in an age-dependent manner.5-HT7, neurogenesis and antidepressants: a promising therapeutic axis for treating depression.Assessing the neuronal serotonergic target-based antidepressant stratagem: impact of in vivo interaction studies and knockout models Sensitization of restraint-induced corticosterone secretion after chronic restraint in rats: involvement of 5-HT₇ receptors.Building a better antipsychotic: receptor targets for the treatment of multiple symptom dimensions of schizophrenia.5-HT(7) receptor modulators: a medicinal chemistry survey of recent patent literature (2004 - 2009).The 5-HT7 receptor as a potential target for treating drug and alcohol abuse.Phe369(7.38) at human 5-HT(7) receptors confers interspecies selectivity to antagonists and partial agonists.Neural mechanisms mediating circadian phase resetting by activation of 5-HT(7) receptors in the dorsal raphe: roles of GABAergic and glutamatergic neurotransmission.Central 5-HT7 receptors are critical for reflex activation of cardiac vagal drive in anaesthetized rats.Homeostatic regulation of sleep in a genetic model of depression in the mouse: effects of muscarinic and 5-HT1A receptor activation.Asenapine modulates mood-related behaviors and 5-HT1A/7 receptors-mediated neurotransmission.Whole genome sequencing of a dizygotic twin suggests a role for the serotonin receptor HTR7 in autism spectrum disorder.

P2860

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P2860

SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

http://www.wikidata.org/entity/Q24672651

description

2003 nî lūn-bûn

@nan

2003 թուականի Յունիսին հրատարակուած գիտական յօդուած

@hyw

2003 թվականի հունիսին հրատարակված գիտական հոդված

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2003年の論文

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2003年論文

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2003年論文

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2003年論文

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2003年論文

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2003年論文

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2003年论文

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name

SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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type

label

SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

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P1433

British Journal of Pharmacology

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SB-656104-A, a novel selective 5-HT7 receptor antagonist, modulates REM sleep in rats

@en

P2093

Alexander J Stevens

http://www.w3.org/2001/XMLSchema#string

Andrew D Gribble

http://www.w3.org/2001/XMLSchema#string

Claire M Scott

http://www.w3.org/2001/XMLSchema#string

David R Thomas

http://www.w3.org/2001/XMLSchema#string

Derek N Middlemiss

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Gary W Price

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Graham Riley

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Ian T Forbes

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Jim J Hagan

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Mario Massagrande

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P2860

Cloning of a novel human serotonin receptor (5-HT7) positively linked to adenylate cyclase

Characterization of [(125)I]-SB-258585 binding to human recombinant and native 5-HT(6) receptors in rat, pig and human brain tissue

5-CT stimulation of adenylyl cyclase activity in guinea-pig hippocampus: evidence for involvement of 5-HT7 and 5-HT1A receptors

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

A novel adenylyl cyclase-activating serotonin receptor (5-HT7) implicated in the regulation of mammalian circadian rhythms

[(3)H]-SB-269970--A selective antagonist radioligand for 5-HT(7) receptors

Functional characterisation of the human cloned 5-HT7 receptor (long form); antagonist profile of SB-258719

Some quantitative uses of drug antagonists

Localization of 5-HT(7) receptors in rat brain by immunocytochemistry, in situ hybridization, and agonist stimulated cFos expression.

A novel, potent, and selective 5-HT(7) antagonist: (R)-3-(2-(2-(4-methylpiperidin-1-yl)ethyl)pyrrolidine-1-sulfonyl) phen ol (SB-269970).

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705-14

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10.1038/SJ.BJP.0705290

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4

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139

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10702710

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12812993

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1573887

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