Structure-activity relationships in a peptidic alpha7 nicotinic acetylcholine receptor antagonist
about
Blockade of neuronal α7-nAChR by α-conotoxin ImI explained by computational scanning and energy calculationsStructural determinants of selective alpha-conotoxin binding to a nicotinic acetylcholine receptor homolog AChBP.A synthetic combinatorial strategy for developing alpha-conotoxin analogs as potent alpha7 nicotinic acetylcholine receptor antagonists.Inhibition of cholinergic pathways in Drosophila melanogaster by α-conotoxins.Structure-activity relationships of alpha-conotoxins targeting neuronal nicotinic acetylcholine receptors.Computational approaches to understand alpha-conotoxin interactions at neuronal nicotinic receptors.Synthetic α-conotoxin mutants as probes for studying nicotinic acetylcholine receptors and in the development of novel drug leads.Acetylcholine promotes binding of α-conotoxin MII at α3 β2 nicotinic acetylcholine receptors.Novel alpha-conotoxins from Conus spurius and the alpha-conotoxin EI share high-affinity potentiation and low-affinity inhibition of nicotinic acetylcholine receptors.Alpha-conotoxins EpI and AuIB switch subtype selectivity and activity in native versus recombinant nicotinic acetylcholine receptors.
P2860
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P2860
Structure-activity relationships in a peptidic alpha7 nicotinic acetylcholine receptor antagonist
description
2000 nî lūn-bûn
@nan
2000 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2000 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
2000年の論文
@ja
2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
name
Structure-activity relationshi ...... tylcholine receptor antagonist
@ast
Structure-activity relationshi ...... tylcholine receptor antagonist
@en
Structure-activity relationshi ...... tylcholine receptor antagonist
@nl
type
label
Structure-activity relationshi ...... tylcholine receptor antagonist
@ast
Structure-activity relationshi ...... tylcholine receptor antagonist
@en
Structure-activity relationshi ...... tylcholine receptor antagonist
@nl
prefLabel
Structure-activity relationshi ...... tylcholine receptor antagonist
@ast
Structure-activity relationshi ...... tylcholine receptor antagonist
@en
Structure-activity relationshi ...... tylcholine receptor antagonist
@nl
P2093
P356
P1476
Structure-activity relationshi ...... tylcholine receptor antagonist
@en
P2093
D E Wemmer
J P Rogers
K Pemberton
P Luginbühl
R C Stevens
P304
P356
10.1006/JMBI.2000.4247
P407
P577
2000-12-15T00:00:00Z