Essential but not vulnerable: indazole sulfonamides targeting inosine monophosphate dehydrogenase as potential leads against Mycobacterium tuberculosis
about
Novel inhibitors of Mycobacterium tuberculosis GuaB2 identified by a target based high-throughput phenotypic screenArpeggio: A Web Server for Calculating and Visualising Interatomic Interactions in Protein StructuresGenomes, structural biology and drug discovery: combating the impacts of mutations in genetic disease and antibiotic resistance.The Bare Essentials of Antibiotic Target Validation.Combating mutations in genetic disease and drug resistance: understanding molecular mechanisms to guide drug design.Targeting DNA Replication and Repair for the Development of Novel Therapeutics against Tuberculosis.Novel Antitubercular 6-Dialkylaminopyrimidine Carboxamides from Phenotypic Whole-Cell High Throughput Screening of a SoftFocus Library: Structure-Activity Relationship and Target Identification Studies.Caught between two proteins: a mycobacterial inhibitor challenges the mold.Mycobacterium tuberculosis Molecular Determinants of Infection, Survival Strategies, and Vulnerable Targets.2-Mercapto-Quinazolinones as Inhibitors of Type II NADH Dehydrogenase and Mycobacterium tuberculosis: Structure-Activity Relationships, Mechanism of Action and Absorption, Distribution, Metabolism, and Excretion Characterization.Expanding benzoxazole based inosine 5'-monophosphate dehydrogenase (IMPDH) inhibitor structure-activity as potential anti-tuberculosis agents.Analysis of a Novel pncA Mutation for Susceptibility to Pyrazinamide Therapy.Fragment-Based Approach to Targeting Inosine-5'-monophosphate Dehydrogenase (IMPDH) from Mycobacterium tuberculosis.Molecular Targets Related Drug Resistance Mechanisms in MDR-, XDR-, and TDR-Mycobacterium tuberculosis Strains.Structural Implications of Mutations Conferring Rifampin Resistance in Mycobacterium leprae.DynaMut: predicting the impact of mutations on protein conformation, flexibility and stability.Understanding molecular consequences of putative drug resistant mutations in Mycobacterium tuberculosisDeath of Mycobacterium tuberculosis by L-arginine starvation
P2860
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P2860
Essential but not vulnerable: indazole sulfonamides targeting inosine monophosphate dehydrogenase as potential leads against Mycobacterium tuberculosis
description
2016 nî lūn-bûn
@nan
2016 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2016 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
name
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@ast
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@en
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@nl
type
label
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@ast
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@en
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@nl
prefLabel
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@ast
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@en
Essential but not vulnerable: ...... nst Mycobacterium tuberculosis
@nl
P2093
P2860
P50
P1476
Essential but Not Vulnerable: ...... nst Mycobacterium tuberculosis
@en
P2093
Alasdair R C Smith
Angela Pacitto
Ardala Breda
Carolyn Selenski
Claire J MacKenzie
Clifton E Barry
Dale J Kempf
Dinakaran Murugesan
Fred Simeons
Gail M Freiberg
P2860
P356
10.1021/ACSINFECDIS.6B00103
P577
2016-10-17T00:00:00Z