Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
about
Small molecule R1498 as a well-tolerated and orally active kinase inhibitor for hepatocellular carcinoma and gastric cancer treatment via targeting angiogenesis and mitosis pathwaysPyrazoles as potential anti-angiogenesis agents: a contemporary overview.Discovery of a highly potent, orally active mitosis/angiogenesis inhibitor r1530 for the treatment of solid tumors.The pyrazolyl-urea GeGe3 inhibits tumor angiogenesis and reveals dystrophia myotonica protein kinase (DMPK)1 as a novel angiogenesis target.
P2860
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
description
2010 nî lūn-bûn
@nan
2010 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@ast
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@en
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@nl
type
label
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@ast
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@en
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@nl
prefLabel
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@ast
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@en
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@nl
P2093
P1476
Pyrazolobenzodiazepines: part I. Synthesis and SAR of a potent class of kinase inhibitors
@en
P2093
Brian Higgins
Christine Lukacs
Chung-Chen Wei
Dorota Miklowski
Fred Konzelmann
Giacomo Pizzolato
Irena Daniewski
P304
P356
10.1016/J.BMCL.2010.08.079
P407
P577
2010-10-15T00:00:00Z