Pyrrolo[1,2-f]triazines as JAK2 inhibitors: achieving potency and selectivity for JAK2 over JAK3
about
Targeted kinase selectivity from kinase profiling data.Selective JAK inhibitors.Discovery of 3H-imidazo[4,5-b]pyridines as potent c-Met kinase inhibitors: design, synthesis, and biological evaluation.Molecular dynamics and integrated pharmacophore-based identification of dual [Formula: see text] inhibitors.Dual inhibitors of Janus kinase 2 and 3 (JAK2/3): designing by pharmacophore- and docking-based virtual screening approach.Ligand-based and e-pharmacophore modeling, 3D-QSAR and hierarchical virtual screening to identify dual inhibitors of spleen tyrosine kinase (Syk) and janus kinase 3 (JAK3).Pharmacophore and docking-based virtual screening approach for the design of new dual inhibitors of Janus kinase 1 and Janus kinase 2.
P2860
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P2860
Pyrrolo[1,2-f]triazines as JAK2 inhibitors: achieving potency and selectivity for JAK2 over JAK3
description
2011 nî lūn-bûn
@nan
2011 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի մարտին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@ast
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@en
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@nl
type
label
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@ast
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@en
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@nl
prefLabel
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@ast
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@en
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@nl
P2093
P1476
Pyrrolo[1,2-f]triazines as JAK ...... selectivity for JAK2 over JAK3
@en
P2093
Arthur V Miller
Ashok V Purandare
George L Trainor
Guifen Zhang
Harold A Mastalerz
Honghe Wan
Javed Khan
Jennifer A Inghrim
John S Sack
P304
P356
10.1016/J.BMCL.2011.01.022
P407
P577
2011-01-11T00:00:00Z