Identification of amides derived from 1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
about
New strategies to maximize therapeutic opportunities for NAMPT inhibitors in oncologyStructural and biochemical analyses of the catalysis and potency impact of inhibitor phosphoribosylation by human nicotinamide phosphoribosyltransferaseStructural basis for resistance to diverse classes of NAMPT inhibitorsPreclinical models of nicotinamide phosphoribosyltransferase inhibitor-mediated hematotoxicity and mitigation by co-treatment with nicotinic acid.Supplementation of nicotinic acid with NAMPT inhibitors results in loss of in vivo efficacy in NAPRT1-deficient tumor models.Crystal structure-based comparison of two NAMPT inhibitors.Cardiotoxicity Associated with Nicotinamide Phosphoribosyltransferase Inhibitors in Rodents and in Rat and Human-Derived Cells Lines.Retinal toxicity, in vivo and in vitro, associated with inhibition of nicotinamide phosphoribosyltransferase.
P2860
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P2860
Identification of amides derived from 1H-pyrazolo[3,4-b]pyridine-5-carboxylic acid as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
description
2013 nî lūn-bûn
@nan
2013 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@ast
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@en
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@nl
type
label
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@ast
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@en
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@nl
prefLabel
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@ast
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@en
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@nl
P2093
P50
P1476
Identification of amides deriv ...... sphoribosyltransferase (NAMPT)
@en
P2093
Alexandre J Buckmelter
Bianca M Liederer
Bingsong Han
Chase C Smith
Deepak Sampath
Dominic J Reynolds
Geeta Sharma
Guangxing Yang
P304
P356
10.1016/J.BMCL.2013.08.074
P407
P577
2013-10-15T00:00:00Z