Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
about
New agents for the treatment of drug-resistant Mycobacterium tuberculosisLearning from the past for TB drug discovery in the futureThe Inosine Monophosphate Dehydrogenase, GuaB2, Is a Vulnerable New Bactericidal Drug Target for Tuberculosis.Target identification by image analysisDesign, synthesis and structure-activity relationship study of wollamide B; a new potential anti TB agent.Recent contributions of structure-based drug design to the development of antibacterial compounds.Conformational Analysis of an Antibacterial Cyclodepsipeptide Active against Mycobacterium tuberculosis by a Combined ROE and RDC Analysis.Antimicrobial Potential of Bacteria Associated with Marine Sea Slugs from North Sulawesi, Indonesia.Color-Coded Super-Resolution Small-Molecule Imaging.New Structural Templates for Clinically Validated and Novel Targets in Antimicrobial Drug Research and Development.StreptomeDB 2.0--an extended resource of natural products produced by streptomycetesIdentification of Thiotetronic Acid Antibiotic Biosynthetic Pathways by Target-directed Genome MiningElucidation of the Teixobactin Pharmacophore.Tailored-pharmacophore model to enhance virtual screening and drug discovery: a case study on the identification of potential inhibitors against drug-resistant Mycobacterium tuberculosis (3R)-hydroxyacyl-ACP dehydratases.Synthetic Cyclic Peptomers as Type III Secretion System Inhibitors.The evolution of genome mining in microbes - a review.Toolbox for Antibiotics Discovery from Microorganisms.Structure of the sliding clamp from the fungal pathogen Aspergillus fumigatus (AfumPCNA) and interactions with Human p21.Strategies for the Discovery and Development of New Antibiotics from Natural Products: Three Case Studies.DNA replication proteins as potential targets for antimicrobials in drug-resistant bacterial pathogens.Recent Advances in Helicobacter pylori Replication: Possible Implications in Adaptation to a Pathogenic Lifestyle and Perspectives for Drug Design.Targeting Phenotypically Tolerant Mycobacterium tuberculosis.DNA Replication in Mycobacterium tuberculosis.Identification of aminopyrimidine-sulfonamides as potent modulators of Wag31-mediated cell elongation in mycobacteria.New structural classes of antituberculosis agents.Kunkel Lecture: Fundamental immunodeficiency and its correction.N-Acetylglucosamine-1-phosphate transferase, WecA, as a validated drug target in Mycobacterium tuberculosis.In vitro and in vivo activity of biapenem against drug-susceptible and rifampicin-resistant Mycobacterium tuberculosis.A Small Covalent Allosteric Inhibitor of Human Cytomegalovirus DNA Polymerase Subunit Interactions.Structural insight into β-Clamp and its interaction with DNA Ligase in Helicobacter pylori.Biosynthesis of methyl-proline containing griselimycins, natural products with anti-tuberculosis activity.Targeting DNA Replication and Repair for the Development of Novel Therapeutics against Tuberculosis.A chemocentric view of the natural product inventory.Caught between two proteins: a mycobacterial inhibitor challenges the mold.New antituberculous drugs derived from natural products: current perspectives and issues in antituberculous drug development.Mycobacterium tuberculosis Molecular Determinants of Infection, Survival Strategies, and Vulnerable Targets.Are highly morphed peptide frameworks lurking silently in microbial genomes valuable as next generation antibiotic scaffolds?Mapping the sequence-structure relationships of simple cyclic hexapeptides.ECBS & ICBS 2015 Joint Meeting: Bringing Chemistry to Life.DNA Replication Fidelity in the Mycobacterium tuberculosis Complex.
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Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
description
2015 nî lūn-bûn
@nan
2015 թուականի Յունիսին հրատարակուած գիտական յօդուած
@hyw
2015 թվականի հունիսին հրատարակված գիտական հոդված
@hy
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
name
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@ast
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@en
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@nl
type
label
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@ast
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@en
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@nl
prefLabel
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@ast
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@en
Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@nl
P2093
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P50
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Antibiotics. Targeting DnaN for tuberculosis therapy using novel griselimycins
@en
P2093
Angela Kling
Armin Bauer
Christine Lair
Claudia König
Deepak V Almeida
Dirk W Heinz
Eric Nuermberger
Evelyne Fontaine
Florence Bordon-Pallier
Gilles Courtemanche
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P304
P3181
P356
10.1126/SCIENCE.AAA4690
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P577
2015-06-01T00:00:00Z