Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities

Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities

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http://www.wikidata.org/entity/Q27703135
Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637)ETS-targeted therapy: can it substitute for MEK inhibitors?Progress in the Development of non-BET Bromodomain Chemical Probes.Bromodomains in Protozoan Parasites: Evolution, Function, and Opportunities for Drug Development.Bromodomain inhibitors and cancer therapy: From structures to applications.Allosteric regulation of epigenetic modifying enzymes.Chemical probes and inhibitors of bromodomains outside the BET family.Regulating the regulators: Epigenetic, transcriptional, and post-translational regulation of RGS proteins.Beyond the BET Family: Targeting CBP/p300 with 4-Acyl Pyrroles.Pharmacophore-based virtual screening, molecular docking, molecular dynamics simulation, and biological evaluation for the discovery of novel BRD4 inhibitors.CREBBP/EP300 bromodomains are critical to sustain the GATA1/MYC regulatory axis in proliferation.An industry perspective on drug target validation
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Transcriptional Profiling of a Selective CREB Binding Protein Bromodomain Inhibitor Highlights Therapeutic Opportunities

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http://www.wikidata.org/entity/Q27703135
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2015 nî lūn-bûn
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2015 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
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2015 թվականի դեկտեմբերին հրատարակված գիտական հոդված
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2015年の論文
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2015年論文
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2015年論文
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2015年論文
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2015年論文
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2015年論文
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2015年论文
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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Transcriptional Profiling of a ...... ghts Therapeutic Opportunities
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10.1016/J.CHEMBIOL.2015.10.013
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