Potentiation of human alpha4beta2 neuronal nicotinic receptors by a Flustra foliacea metabolite
about
Allosteric modulator Desformylflustrabromine relieves the inhibition of α2β2 and α4β2 nicotinic acetylcholine receptors by β-amyloid(1-42) peptideSynthesis of desformylflustrabromine and its evaluation as an alpha4beta2 and alpha7 nACh receptor modulatorUnravelling the mechanism of action of NS9283, a positive allosteric modulator of (α4)3(β2)2 nicotinic ACh receptorsDeconstruction of the α4β2 nicotinic acetylcholine receptor positive allosteric modulator desformylflustrabromineOrthosteric and Allosteric Ligands of Nicotinic Acetylcholine Receptors for Smoking CessationMarine Indole AlkaloidsTargeting α4β2 nicotinic acetylcholine receptors in central nervous system disorders: perspectives on positive allosteric modulation as a therapeutic approach.Pharmacological characterization of the allosteric modulator desformylflustrabromine and its interaction with alpha4beta2 neuronal nicotinic acetylcholine receptor orthosteric ligands.Structural answers and persistent questions about how nicotinic receptors work.Allosteric modulators of the α4β2 subtype of neuronal nicotinic acetylcholine receptors.Positive allosteric modulators as an approach to nicotinic acetylcholine receptor-targeted therapeutics: advantages and limitations.Desformylflustrabromine (dFBr) and [3H]dFBr-Labeled Binding Sites in a Nicotinic Acetylcholine Receptor.Marine AChE inhibitors isolated from Geodia barretti: natural compounds and their synthetic analogs.Desformylflustrabromine Modulates α4β2 Neuronal Nicotinic Acetylcholine Receptor High- and Low-Sensitivity Isoforms at Allosteric Clefts Containing the β2 SubunitPhotolabeling a Nicotinic Acetylcholine Receptor (nAChR) with an (α4)3(β2)2 nAChR-Selective Positive Allosteric Modulator.Allosteric modulation of alpha4beta2 nicotinic acetylcholine receptors by HEPESPositive allosteric modulation of α4β2 nicotinic acetylcholine receptors as a new approach to smoking reduction: evidence from a rat model of nicotine self-administration.Recent progress in neuroactive marine natural products.Doubly prenylated tryptamines: cytotoxicity, antimicrobial activity and cyclisation to the marine natural product flustramine A.Effects of nicotine in combination with drugs described as positive allosteric nicotinic acetylcholine receptor modulators in vitro: discriminative stimulus and hypothermic effects in mice.Levamisole: A Positive Allosteric Modulator for the α3β4 Nicotinic Acetylcholine Receptors Prevents Weight Gain in the CD-1 Mice on a High Fat Diet.Nicotinic acetylcholine receptors in neuropathic and inflammatory pain.LY2087101 and dFBr share transmembrane binding sites in the (α4)3(β2)2 Nicotinic Acetylcholine Receptor.Role of the Cys Loop and Transmembrane Domain in the Allosteric Modulation of α4β2 Nicotinic Acetylcholine Receptors.Unraveling amino acid residues critical for allosteric potentiation of (α4)3(β2)2-type nicotinic acetylcholine receptor responses.
P2860
Q24629740-9D8A8B0D-D4BE-4D19-B4CF-A8F306BC7F8CQ24632272-3705ABCA-E6FF-41BA-A866-F70DC3AA7623Q24634426-C2688BED-895E-4A65-99DC-D534018FA4D1Q24634672-26C25AA8-9849-4C2E-8A20-E77907BD0489Q26774830-62C3688B-2342-4226-9B21-D6F2CD8FDA62Q26796630-9ED9FC0B-19E7-4AD5-98F1-5120B83AD8A2Q27693356-AC31A041-C638-48A5-961F-B420D967CEEEQ34128766-6E4218E6-E3F0-446A-A1AD-5974271A28EFQ34782188-40193310-6CC6-4CC8-96F6-F30A454C93E1Q35182101-D6EED878-95F4-4191-9097-F5BFB6FD02DFQ35182164-D4135DA8-C154-462D-AB72-B1A6AB273B86Q35745950-756B2A74-80CF-4F1B-ABC9-F2EB4C788A9FQ35875939-A9DEEB22-1091-4324-AFF3-AF103EAD9D43Q35897805-8A28D798-3052-4EB4-BA11-2CCA7AF6BE47Q36852497-3A484E39-CF3B-43A4-AA08-48159D302E96Q37117186-1915D331-BBC7-4F31-902F-3D13269DB8C2Q37230901-92EAE51F-6F0B-4983-A0EF-AB0F0C3CD2E1Q37639029-727D9FD4-0CE1-489C-AED8-4EB446B2294DQ39113781-04864F23-2C86-4368-A629-C423C7F10825Q42365798-207542F0-0A13-4529-A888-C92A1913C0C8Q47177367-A3C11B72-095C-49EC-8ED7-18C05E725140Q47739924-F2B07FBE-3AEE-4BB1-A0DA-2953D3EDB131Q48204150-16F57A0C-0A91-4346-9569-04F7C32CF08CQ48213996-BEDE7B45-68B4-4A34-83E1-04C21278B2C8Q48522591-D941BEBF-3CE7-4CE3-940E-0CCCB3BDD937
P2860
Potentiation of human alpha4beta2 neuronal nicotinic receptors by a Flustra foliacea metabolite
description
2005 nî lūn-bûn
@nan
2005 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2005 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2005年の論文
@ja
2005年論文
@yue
2005年論文
@zh-hant
2005年論文
@zh-hk
2005年論文
@zh-mo
2005年論文
@zh-tw
2005年论文
@wuu
name
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@ast
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@en
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@nl
type
label
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@ast
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@en
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@nl
prefLabel
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@ast
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@en
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@nl
P2093
P1433
P1476
Potentiation of human alpha4be ...... a Flustra foliacea metabolite
@en
P2093
Francisco Sala
Gabriele M König
José Antonio Bernal
José Mulet
Krishna P Reddy
Lars Peters
Manuel Criado
Philip Wikman
Salvador Sala
P304
P356
10.1016/J.NEULET.2004.10.002
P407
P577
2005-01-01T00:00:00Z