Molecular basis for the species selectivity of the neurokinin-1 receptor antagonists CP-96,345 and RP67580
about
Hydrophilic side chains in the third and seventh transmembrane helical domains of human A2A adenosine receptors are required for ligand recognitionThe Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsThe C9 methyl group of retinal interacts with glycine-121 in rhodopsin.Genetic and pharmacological disruption of neurokinin 1 receptor function decreases anxiety-related behaviors and increases serotonergic function.[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.Quantification of central substance P receptor occupancy by aprepitant using small animal positron emission tomography.Molecular Architecture of G Protein-Coupled Receptors.Distribution and pharmacological characterization of primate NK-1 and NK-3 tachykinin receptors in the central nervous system of the rhesus monkey.Central versus peripheral site of action of the tachykinin NK1-antagonist RP 67580 in inhibiting chemonociception.Mechanical Conflict System: A Novel Operant Method for the Assessment of Nociceptive Behavior.The molecular basis for high affinity of a universal ligand for human bombesin receptor (BnR) family members.Potentiation of brain stimulation reward by morphine: effects of neurokinin-1 receptor antagonism.Two nonpeptide tachykinin antagonists act through epitopes on corresponding segments of the NK1 and NK2 receptors.Relationships between neurokinin receptor-expressing interstitial cells of Cajal and tachykininergic nerves in the gut.Construction of a novel bifunctional biogenic amine receptor by two point mutations of the H2-histamine receptorMolecular basis for the selectivity of the mammalian bombesin peptide, neuromedin B, for its receptorAntinociceptive activity of NK1 receptor antagonists: non-specific effects of racemic RP67580.Differences in the effects of NK1-receptor antagonists, (+/-)-CP 96,345 and CP 99,994, on agonist-induced responses in guinea-pig trachea.Characterization of NK1 and NK2 tachykinin receptors in guinea-pig and rat bronchopulmonary and vascular systems.Comparison of tachykinin NK1 and NK2 receptors in the circular muscle of the guinea-pig ileum and proximal colon.Tachykinin NK1 receptor subtypes in the rat urinary bladder.
P2860
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P2860
Molecular basis for the species selectivity of the neurokinin-1 receptor antagonists CP-96,345 and RP67580
description
1992 nî lūn-bûn
@nan
1992 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1992 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
1992年の論文
@ja
1992年論文
@yue
1992年論文
@zh-hant
1992年論文
@zh-hk
1992年論文
@zh-mo
1992年論文
@zh-tw
1992年论文
@wuu
name
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@ast
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@en
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@nl
type
label
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@ast
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@en
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@nl
prefLabel
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@ast
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@en
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@nl
P2093
P1476
Molecular basis for the specie ...... agonists CP-96,345 and RP67580
@en
P2093
P304
P407
P577
1992-12-25T00:00:00Z