[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain. - Wikidata - awgldk - TriplyDB

[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

http://www.wikidata.org/entity/Q35100845

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Anxiolytic-like effects of the neurokinin 1 receptor antagonist GR-205171 in the elevated plus maze and contextual fear-potentiated startle model of anxiety in gerbils.PET imaging of neurokinin-1 receptors with [(18)F]SPA-RQ in human subjects: assessment of reference tissue models and their test-retest reproducibility.A pharmacokinetic PET study of NK₁ receptor occupancy.First evaluation of [11C]R116301 as an in vivo tracer of NK1 receptors in man Increased neurokinin-1 receptor availability in the amygdala in social anxiety disorder: a positron emission tomography study with [11C]GR205171.Considerations in the Development of Reversibly Binding PET Radioligands for Brain Imaging.Neurokinin-1 receptor antagonist orvepitant is an effective inhibitor of itch-associated response in a Mongolian gerbil model of scratching behaviour.Differential effects of aprepitant, a clinically used neurokinin-1 receptor antagonist on the expression of conditioned psychostimulant versus opioid reward.Association between amygdala neurokinin-1 receptor availability and anxiety-related personality traits

P2860

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P2860

[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

http://www.wikidata.org/entity/Q35100845

description

2006 nî lūn-bûn

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2006 թուականի Մայիսին հրատարակուած գիտական յօդուած

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2006 թվականի մայիսին հրատարակված գիտական հոդված

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2006年の論文

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2006年学术文章

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2006年学术文章

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2006年学术文章

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2006年学术文章

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2006年学术文章

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2006年學術文章

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name

[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

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[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

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type

label

[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

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[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

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prefLabel

[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

@ast

[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

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British Journal of Pharmacology

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[3H]GR205171 displays similar NK1 receptor binding profile in gerbil and human brain.

@en

P2093

Cristiana Griffante

http://www.w3.org/2001/XMLSchema#string

Filippo Andreetta

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Mauro Corsi

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Renzo Carletti

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P2860

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

The tachykinin NK1 receptor in the brain: pharmacology and putative functions

The gerbil elevated plus-maze II: anxiolytic-like effects of selective neurokinin NK1 receptor antagonists

The antidepressant-like effects of neurokinin NK1 receptor antagonists in a gerbil tail suspension test

Distinct mechanism for antidepressant activity by blockade of central substance P receptors

Molecular basis for the species selectivity of the neurokinin-1 receptor antagonists CP-96,345 and RP67580

Comparison of the functional blockade of rat substance P (NK1) receptors by GR205171, RP67580, SR140333 and NKP-608.

GR205171: a novel antagonist with high affinity for the tachykinin NK1 receptor, and potent broad-spectrum anti-emetic activity.

Substance P receptor antagonists in psychiatry: rationale for development and therapeutic potential.

L-733,060, a novel tachykinin NK1 receptor antagonist; effects in [Ca2+]i mobilisation, cardiovascular and dural extravasation assays.

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39-45

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10.1038/SJ.BJP.0706697

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1

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7275187

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16501582

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1617048

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