[3H]-LY341495 as a novel antagonist radioligand for group II metabotropic glutamate (mGlu) receptors: characterization of binding to membranes of mGlu receptor subtype expressing cells
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Distinct roles of metabotropic glutamate receptor dimerization in agonist activation and G-protein couplingThe mGluR2 positive allosteric modulator BINA decreases cocaine self-administration and cue-induced cocaine-seeking and counteracts cocaine-induced enhancement of brain reward function in ratsCharacterization of an mGluR2/3 negative allosteric modulator in rodent models of depressionThe mGluR2 positive allosteric modulator, SAR218645, improves memory and attention deficits in translational models of cognitive symptoms associated with schizophreniaN-methyl-D-aspartate receptors and large conductance calcium-sensitive potassium channels inhibit the release of opioid peptides that induce mu-opioid receptor internalization in the rat spinal cord.Pharmacological reversal of synaptic plasticity deficits in the mouse model of fragile X syndrome by group II mGluR antagonist or lithium treatment.Cerebral 5-HT2A receptor binding, but not mGluR2, is increased in tryptophan hydroxylase 2 decrease-of-function micePharmacological blockade of group II metabotropic glutamate receptors reduces the growth of glioma cells in vivo.Progress toward advanced understanding of metabotropic glutamate receptors: structure, signaling and therapeutic indicationsGroup II/III metabotropic glutamate receptors exert endogenous activity-dependent modulation of TRPV1 receptors on peripheral nociceptorsType 2 metabotropic glutamate receptor (mGluR2) fails to negatively couple to cGMP in stably transfected cells.Long-term depression at parallel fiber to Golgi cell synapses.Actions of LY341495 on metabotropic glutamate receptor-mediated responses in the neonatal rat spinal cord.Involvement of metabotropic glutamate receptors in excitatory amino acid and GABA release following spinal cord injury in rat.Developmental decrease in synaptic facilitation at the mouse hippocampal mossy fibre synapse.New type of synaptically mediated epileptiform activity independent of known glutamate and GABA receptors.The peptidic antidepressant spadin interacts with prefrontal 5-HT(4) and mGluR(2) receptors in the control of serotonergic function.Synthesis and Preliminary Studies of a Novel Negative Allosteric Modulator, 7-((2,5-Dioxopyrrolidin-1-yl)methyl)-4-(2-fluoro-4-[11C]methoxyphenyl) quinoline-2-carboxamide, for Imaging of Metabotropic Glutamate Receptor 2.NAD(P)H fluorescence transients after synaptic activity in brain slices: predominant role of mitochondrial function.A group II metabotropic glutamate receptor 3 (mGlu3, GRM3) isoform implicated in schizophrenia interacts with canonical mGlu3 and reduces ligand binding.Increased metabotropic glutamate 2/3 receptor binding in the perigenual anterior cingulate cortex of Cloninger type 2 alcoholics: a whole-hemisphere autoradiography study.Oligomerization of a G protein-coupled receptor in neurons controlled by its structural dynamics.
P2860
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P2860
[3H]-LY341495 as a novel antagonist radioligand for group II metabotropic glutamate (mGlu) receptors: characterization of binding to membranes of mGlu receptor subtype expressing cells
description
1999 nî lūn-bûn
@nan
1999 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1999 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
1999年の論文
@ja
1999年論文
@yue
1999年論文
@zh-hant
1999年論文
@zh-hk
1999年論文
@zh-mo
1999年論文
@zh-tw
1999年论文
@wuu
name
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@ast
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@en
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@nl
type
label
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@ast
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@en
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@nl
prefLabel
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@ast
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@en
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@nl
P2093
P3181
P1433
P1476
[3H]-LY341495 as a novel antag ...... eptor subtype expressing cells
@en
P2093
B G Johnson
D D Schoepp
M B Arnold
P L Ornstein
R A Wright
W J Wheeler
P304
P3181
P356
10.1016/S0028-3908(99)00053-2
P407
P577
1999-10-01T00:00:00Z