{Beta}-blocker drugs mediate calcium signaling in native central nervous system neurons by {beta}-arrestin-biased agonism
about
Ligand-specific endocytic dwell times control functional selectivity of the cannabinoid receptor 1The β-blocker Nebivolol Is a GRK/β-arrestin biased agonistMedicinal chemistry for 2020Induction of cardiac fibrosis by β-blocker in G protein-independent and G protein-coupled receptor kinase 5/β-arrestin2-dependent Signaling pathways.The C57BL/6 genetic background confers cardioprotection in iron-overloaded miceMechanisms of Biased β-Arrestin-Mediated Signaling Downstream from the Cannabinoid 1 Receptor.Achievement of a target dose of bisoprolol may not be a preferred option for attenuating pressure overload-induced cardiac hypertrophy and fibrosisAKAP-dependent modulation of BCAM/Lu adhesion on normal and sickle cell disease RBCs revealed by force nanoscopy.Insights into the structural biology of G-protein coupled receptors impacts drug design for central nervous system neurodegenerative processes.The Multiple Waves of Cannabinoid 1 Receptor Signaling.β-adrenergic signaling broadly contributes to LTP induction.Imaging GPCRs trafficking and signaling with total internal reflection fluorescence microscopy in cultured neuronsDivergent agonist selectivity in activating β1- and β2-adrenoceptors for G-protein and arrestin coupling.
P2860
Q28245037-706F3DAF-A457-4CEF-BE45-DF19D3CF7DFEQ34972784-77F669DD-D938-4642-BCCD-E83B1598411FQ35593223-1E9667F9-A0F6-42D8-94BC-5568B646BBB4Q36318886-141307DC-7F45-470E-AD1D-0E0A1097306AQ36569080-1019905F-0BAB-4750-B27D-9D8972F2F42CQ36947742-EDEBB66D-264A-4E23-B9AE-3400B4A409C4Q37288326-A20FA5A9-4162-4CFE-83C9-BF931F80387FQ37700189-98B90B16-5A05-436C-8932-14A2589BEC43Q38247995-73BA1EFE-AFFB-4AA5-9498-9BD865795DBCQ38874828-C41CDEA2-FDA5-425B-BF8A-5056B94910ECQ41282699-7697DC2F-186C-4B8D-A261-6BF3DBA845E3Q42285998-B79C8947-59D0-4E7E-9C34-A6A4F05BE9EAQ45227106-8BD11E8A-C53E-49AA-A686-E3C4C26C897F
P2860
{Beta}-blocker drugs mediate calcium signaling in native central nervous system neurons by {beta}-arrestin-biased agonism
description
2010 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
article publié dans les Procee ...... f the United States of America
@fr
artículu científicu espublizáu en 2010
@ast
im Dezember 2010 veröffentlichter wissenschaftlicher Artikel
@de
scientific journal article
@en
vedecký článok (publikovaný 2010/12/07)
@sk
vědecký článek publikovaný v roce 2010
@cs
wetenschappelijk artikel (gepubliceerd op 2010/12/07)
@nl
наукова стаття, опублікована в грудні 2010
@uk
name
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@ast
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@en
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@nl
type
label
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@ast
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@en
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@nl
prefLabel
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@ast
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@en
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@nl
P2860
P3181
P356
P1476
{Beta}-blocker drugs mediate c ...... {beta}-arrestin-biased agonism
@en
P2093
Anastassios V. Tzingounis
P2860
P304
21028–21033
P3181
P356
10.1073/PNAS.1004169107
P407
P577
2010-12-07T00:00:00Z