Unravelling intrinsic efficacy and ligand bias at G protein coupled receptors: A practical guide to assessing functional data.
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Functional Characterization of a Novel Series of Biased Signaling Dopamine D3 Receptor Agonists.Functional selectivity at G-protein coupled receptors: Advancing cannabinoid receptors as drug targets.The synthetic cannabinoid WIN55,212-2 mesylate decreases the production of inflammatory mediators in rheumatoid arthritis synovial fibroblasts by activating CB2, TRPV1, TRPA1 and yet unidentified receptor targets.Modulation of opioid receptor affinity and efficacy via N-substitution of 9β-hydroxy-5-(3-hydroxyphenyl)morphan: Synthesis and computer simulation study.A single extracellular amino acid in Free Fatty Acid Receptor 2 defines antagonist species selectivity and G protein selection bias.Modelling and simulation of biased agonism dynamics at a G protein-coupled receptor.Methodical Challenges and a Possible Resolution in the Assessment of Receptor Reserve for Adenosine, an Agonist with Short Half-Life.Measuring ligand efficacy at the mu-opioid receptor using a conformational biosensorCurrent Concepts and Treatments of Schizophrenia
P2860
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P2860
Unravelling intrinsic efficacy and ligand bias at G protein coupled receptors: A practical guide to assessing functional data.
description
2015 nî lūn-bûn
@nan
2015 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2015 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2015年の論文
@ja
2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
@wuu
name
Unravelling intrinsic efficacy ...... to assessing functional data.
@ast
Unravelling intrinsic efficacy ...... to assessing functional data.
@en
type
label
Unravelling intrinsic efficacy ...... to assessing functional data.
@ast
Unravelling intrinsic efficacy ...... to assessing functional data.
@en
prefLabel
Unravelling intrinsic efficacy ...... to assessing functional data.
@ast
Unravelling intrinsic efficacy ...... to assessing functional data.
@en
P2093
P50
P1476
Unravelling intrinsic efficacy ...... to assessing functional data.
@en
P2093
David A Hall
Lisa A Stott
Nicholas D Holliday
P356
10.1016/J.BCP.2015.10.011
P407
P577
2015-10-15T00:00:00Z