Inverse agonist activity at the alpha(2A)-adrenergic receptor.
about
Enhanced spontaneous activity of the mu opioid receptor by cysteine mutations: characterization of a tool for inverse agonist screeningComputationally-predicted CB1 cannabinoid receptor mutants show distinct patterns of salt-bridges that correlate with their level of constitutive activity reflected in G protein coupling levels, thermal stability, and ligand binding.Changes in postnatal norepinephrine alter alpha-2 adrenergic receptor development.Inverse agonism and its therapeutic significance.(4-(Bis(4-fluorophenyl)methyl)piperazin-1-yl)(cyclohexyl)methanone hydrochloride (LDK1229): a new cannabinoid CB1 receptor inverse agonist from the class of benzhydryl piperazine analogs.Recent advances in drug action and therapeutics: relevance of novel concepts in G-protein-coupled receptor and signal transduction pharmacology.Alpha2-adrenoceptor action on cell proliferation and mammary tumour growth in miceAgonist binding, agonist affinity and agonist efficacy at G protein-coupled receptorsMapping the structural requirements in the CB1 cannabinoid receptor transmembrane helix II for signal transductionEffects in vitro and in vivo by apomorphine in the rat corpus cavernosum.Mechanisms of inverse agonist action at D2 dopamine receptors.Suppression of osteoclastogenesis via α2-adrenergic receptors.
P2860
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P2860
Inverse agonist activity at the alpha(2A)-adrenergic receptor.
description
2001 nî lūn-bûn
@nan
2001 թուականի Մարտին հրատարակուած գիտական յօդուած
@hyw
2001 թվականի մարտին հրատարակված գիտական հոդված
@hy
2001年の論文
@ja
2001年論文
@yue
2001年論文
@zh-hant
2001年論文
@zh-hk
2001年論文
@zh-mo
2001年論文
@zh-tw
2001年论文
@wuu
name
Inverse agonist activity at the alpha(2A)-adrenergic receptor.
@ast
Inverse agonist activity at the alpha(2A)-adrenergic receptor.
@en
type
label
Inverse agonist activity at the alpha(2A)-adrenergic receptor.
@ast
Inverse agonist activity at the alpha(2A)-adrenergic receptor.
@en
prefLabel
Inverse agonist activity at the alpha(2A)-adrenergic receptor.
@ast
Inverse agonist activity at the alpha(2A)-adrenergic receptor.
@en
P2093
P356
P1476
Inverse agonist activity at the alpha(2A)-adrenergic receptor
@en
P2093
P304
P356
10.1124/MOL.59.3.532
P50
P577
2001-03-01T00:00:00Z