Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry.
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Early cerebral activities of the environmental estrogen bisphenol A appear to act via the somatostatin receptor subtype sst(2)Stepping into the omics era: Opportunities and challenges for biomaterials science and engineeringIdentification of multiple somatostatin receptors in the rat somatosensory cortex during developmentSomatostatin inhibits cell migration and reduces cell counts of human keratinocytes and delays epidermal wound healing in an ex vivo wound modelThe Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsLibrary design concepts and implementation strategies.Automated ARGET ATRP Accelerates Catalyst Optimization for the Synthesis of Thiol-Functionalized Polymers.Combinatorial target-guided ligand assembly: identification of potent subtype-selective c-Src inhibitors.Homo- and heterodimerization of somatostatin receptor subtypes. Inactivation of sst(3) receptor function by heterodimerization with sst(2A).Chemical genetics: ligand-based discovery of gene function.Medical treatment of diabetic retinopathy with somatostatin analogues.Fabrication of combinatorial polymer scaffold libraries.X-ray imaging optimization of 3D tissue engineering scaffolds via combinatorial fabrication methods.Conformationally homogeneous heterocyclic pseudotetrapeptides as three-dimensional scaffolds for rational drug design: receptor-selective somatostatin analogues.Regulation of somatostatin receptor 4-mediated cytostatic effects by CD26 in malignant pleural mesotheliomaCombinatorial and high-throughput screening of biomaterials.Brain somatostatin: a candidate inhibitory role in seizures and epileptogenesis.Peptide interactions with G-protein coupled receptors.Somatostatin analogs and radiopeptides in cancer therapy.Pharmacological rationale for the use of somatostatin and analogues in portal hypertension.SST3-selective potent peptidic somatostatin receptor antagonists.Homologous and heterologous in vitro regulation of pituitary receptors for somatostatin, growth hormone (GH)-releasing hormone, and ghrelin in a nonhuman primate (Papio anubis).Somatostatin analogs: a new tool for the management of Graves' ophthalmopathy.Treatment of endocrine pancreatic tumors.Recent developments in the therapy of acromegaly.Modification of ghrelin receptor signaling by somatostatin receptor-5 regulates insulin release.Peptide receptor targeting in cancer: the somatostatin paradigm.Selective agonism in somatostatin receptor signaling and regulation.Involvement of somatostatin receptor subtypes in membrane ion channel modification by somatostatin in pituitary somatotropes.Biology and treatment of metastatic gastrointestinal neuroendocrine tumors.Inhibitory effect of somatostatin-14 on L-type voltage-gated calcium channels in cultured cone photoreceptors requires intracellular calciumThe somatostatin receptor subtype 5 in neuroendocrine tumours.Anticonvulsant neuropeptides as drug leads for neurological diseases.High-throughput rheology in a microfluidic device.Improvement of drug-like properties of peptides: the somatostatin paradigm.Heterodimerization of β2 adrenergic receptor and somatostatin receptor 5: Implications in modulation of signaling pathway.The recent progress in proteochemometric modelling: focusing on target descriptors, cross-term descriptors and application scope.Cell growth inhibition and functioning of human somatostatin receptor type 2 are modulated by receptor heterodimerization.Somatostatin decreases voltage-gated Ca2+ currents in GH3 cells through activation of somatostatin receptor 2.Expression of somatostatin receptors in normal and cirrhotic human liver and in hepatocellular carcinoma.
P2860
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P2860
Rapid identification of subtype-selective agonists of the somatostatin receptor through combinatorial chemistry.
description
1998 nî lūn-bûn
@nan
1998 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1998 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
1998年の論文
@ja
1998年論文
@yue
1998年論文
@zh-hant
1998年論文
@zh-hk
1998年論文
@zh-mo
1998年論文
@zh-tw
1998年论文
@wuu
name
Rapid identification of subtyp ...... rough combinatorial chemistry.
@ast
Rapid identification of subtyp ...... rough combinatorial chemistry.
@en
type
label
Rapid identification of subtyp ...... rough combinatorial chemistry.
@ast
Rapid identification of subtyp ...... rough combinatorial chemistry.
@en
prefLabel
Rapid identification of subtyp ...... rough combinatorial chemistry.
@ast
Rapid identification of subtyp ...... rough combinatorial chemistry.
@en
P2093
P1433
P1476
Rapid identification of subtyp ...... rough combinatorial chemistry.
@en
P2093
Chapman KT
Degrado SJ
Hutchins SM
P304
P356
10.1126/SCIENCE.282.5389.737
P407
P577
1998-10-01T00:00:00Z