Inhibition of the complete set of mammalian secreted phospholipases A(2) by indole analogues: a structure-guided study.

Inhibition of the complete set of mammalian secreted phospholipases A(2) by indole analogues: a structure-guided study.

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http://www.wikidata.org/entity/Q33199743
Blockade of human group X secreted phospholipase A2 (GX-sPLA2)-induced airway inflammation and hyperresponsiveness in a mouse asthma model by a selective GX-sPLA2 inhibitorInhibition of lipoprotein-associated phospholipase A2 reduces complex coronary atherosclerotic plaque developmentPhospholipase A2 enzymes: physical structure, biological function, disease implication, chemical inhibition, and therapeutic interventionHighly specific and broadly potent inhibitors of mammalian secreted phospholipases A2Inhibition of secreted phospholipases A₂ by 2-oxoamides based on α-amino acids: Synthesis, in vitro evaluation and molecular docking calculations.In vitro anti-Plasmodium falciparum properties of the full set of human secreted phospholipases A2.Biochemical characterization of selective inhibitors of human group IIA secreted phospholipase A(2) and hyaluronic acid-linked inhibitor conjugates.Neuroprotective effects of a nanocrystal formulation of sPLA(2) inhibitor PX-18 in cerebral ischemia/reperfusion in gerbilsDevelopment of a potent 2-oxoamide inhibitor of secreted phospholipase A2 guided by molecular docking calculations and molecular dynamics simulations.Structural basis for functional selectivity and ligand recognition revealed by crystal structures of human secreted phospholipase A2 group IIE.A novel phospholipase A2 (D49) from the venom of the Crotalus oreganus abyssus (North American Grand canyon rattlesnake).The first potent inhibitor of mammalian group X secreted phospholipase A2: elucidation of sites for enhanced bindingHigh plasma phospholipase A2 activity, inflammation markers, and LDL alterations in obesity with or without type 2 diabetes.Formamidine hydrochloride as an amino surrogate: I2-catalyzed oxidative amidation of aryl methyl ketones leading to free (N-H) α-ketoamides.pCRP-mCRP Dissociation Mechanisms as Potential Targets for the Development of Small-Molecule Anti-Inflammatory Chemotherapeutics.
P2860

Inhibition of the complete set of mammalian secreted phospholipases A(2) by indole analogues: a structure-guided study.

Item
http://www.wikidata.org/entity/Q33199743
description
2004 nî lūn-bûn
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2004 թուականի Ապրիլին հրատարակուած գիտական յօդուած
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2004 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2004年の論文
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2004年論文
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2004年論文
@zh-hant
2004年論文
@zh-hk
2004年論文
@zh-mo
2004年論文
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2004年论文
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name
Inhibition of the complete set ...... ues: a structure-guided study.
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Inhibition of the complete set ...... ues: a structure-guided study.
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type
label
Inhibition of the complete set ...... ues: a structure-guided study.
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Inhibition of the complete set ...... ues: a structure-guided study.
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prefLabel
Inhibition of the complete set ...... ues: a structure-guided study.
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Inhibition of the complete set ...... ues: a structure-guided study.
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Inhibition of the complete set ...... ues: a structure-guided study.
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P2093
P304
P31
P356
P407
P433
P478
P50
P577
P5875
P698