New chemical scaffolds for human african trypanosomiasis lead discovery from a screen of tyrosine kinase inhibitor drugs
about
Kinases as druggable targets in trypanosomatid protozoan parasitesDiscovery of a Carbazole-Derived Lead Drug for Human African TrypanosomiasisAn overview of travel-associated central nervous system infectious diseases: risk assessment, general considerations and future directions.EVALUATION OF AROMATIC 6-SUBSTITUTED THIENOPYRIMIDINES AS SCAFFOLDS AGAINST PARASITES THAT CAUSE TRYPANOSOMIASIS, LEISHMANIASIS, AND MALARIA.Identification of "Preferred" Human Kinase Inhibitors for Sleeping Sickness Lead Discovery. Are Some Kinases Better than Others for Inhibitor Repurposing?Repurposing strategies for tropical disease drug discovery.Glycogen Synthase Kinase 3β Promotes the Endocytosis of Transferrin in the African TrypanosomeEmerging therapies: angiogenesis inhibitors for ovarian cancer.Repurposing of Human Kinase Inhibitors in Neglected Protozoan Diseases.Novel Effects of Lapatinib Revealed in the African Trypanosome by Using Hypothesis-Generating Proteomics and Chemical Biology Strategies.AEE788 Inhibits Basal Body Assembly and Blocks DNA Replication in the African Trypanosome.Optimization of physicochemical properties for 4-anilinoquinazoline inhibitors of trypanosome proliferation.Series of Alkynyl-Substituted Thienopyrimidines as Inhibitors of Protozoan Parasite ProliferationNovel lead compounds in pre-clinical development against African sleeping sickness
P2860
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P2860
New chemical scaffolds for human african trypanosomiasis lead discovery from a screen of tyrosine kinase inhibitor drugs
description
2014 nî lūn-bûn
@nan
2014 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի հունվարին հրատարակված գիտական հոդված
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2014年の論文
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2014年学术文章
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2014年学术文章
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2014年学术文章
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2014年学术文章
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2014年学术文章
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2014年學術文章
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name
New chemical scaffolds for hum ...... yrosine kinase inhibitor drugs
@ast
New chemical scaffolds for hum ...... yrosine kinase inhibitor drugs
@en
type
label
New chemical scaffolds for hum ...... yrosine kinase inhibitor drugs
@ast
New chemical scaffolds for hum ...... yrosine kinase inhibitor drugs
@en
prefLabel
New chemical scaffolds for hum ...... yrosine kinase inhibitor drugs
@ast
New chemical scaffolds for hum ...... yrosine kinase inhibitor drugs
@en
P2093
P2860
P356
P1476
New chemical scaffolds for hum ...... yrosine kinase inhibitor drugs
@en
P2093
Kojo Mensa-Wilmot
Ranjan Behera
Sarah M Thomas
P2860
P304
P356
10.1128/AAC.01691-13
P407
P577
2014-01-27T00:00:00Z