Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions
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Adding Molecules to Food, Pros and Cons: A Review on Synthetic and Natural Food AdditivesAllosteric modulation of purine and pyrimidine receptors.Allosteric interactions across native adenosine-A3 receptor homodimers: quantification using single-cell ligand-binding kinetics.The A3 adenosine receptor as multifaceted therapeutic target: pharmacology, medicinal chemistry, and in silico approaches.Therapeutic potential of A2 and A3 adenosine receptor: a review of novel patented ligands.Allosteric interactions at adenosine A(1) and A(3) receptors: new insights into the role of small molecules and receptor dimerization.Biophysical Detection of Diversity and Bias in GPCR Function.Synthesis and characterization of high-affinity 4,4-difluoro-4-bora-3a,4a-diaza-s-indacene-labeled fluorescent ligands for human β-adrenoceptors.Negative cooperativity across β1-adrenoceptor homodimers provides insights into the nature of the secondary low-affinity CGP 12177 β1-adrenoceptor binding conformation.Kinetic analysis of antagonist-occupied adenosine-A3 receptors within membrane microdomains of individual cells provides evidence of receptor dimerization and allosterism.Synthesis of BODIPY derivatives substituted with various bioconjugatable linker groups: a construction kit for fluorescent labeling of receptor ligands.
P2860
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P2860
Antagonist selective modulation of adenosine A1 and A3 receptor pharmacology by the food dye Brilliant Black BN: evidence for allosteric interactions
description
2010 nî lūn-bûn
@nan
2010 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Antagonist selective modulatio ...... ce for allosteric interactions
@ast
Antagonist selective modulatio ...... ce for allosteric interactions
@en
type
label
Antagonist selective modulatio ...... ce for allosteric interactions
@ast
Antagonist selective modulatio ...... ce for allosteric interactions
@en
prefLabel
Antagonist selective modulatio ...... ce for allosteric interactions
@ast
Antagonist selective modulatio ...... ce for allosteric interactions
@en
P2860
P356
P1476
Antagonist selective modulatio ...... ce for allosteric interactions
@en
P2093
P2860
P304
P356
10.1124/MOL.109.063065
P577
2010-01-19T00:00:00Z