3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
about
Design and synthesis of novel xyloketal derivatives and their protective activities against H2O2-induced HUVEC injury.Novologues containing a benzamide side chain manifest anti-proliferative activity against two breast cancer cell lines.Activation of Hsp90 Enzymatic Activity and Conformational Dynamics through Rationally Designed Allosteric Ligands.Identification of a new scaffold for hsp90 C-terminal inhibitionDesign, synthesis and biological evaluation of biphenylamide derivatives as Hsp90 C-terminal inhibitorsExploiting conformational dynamics in drug discovery: design of C-terminal inhibitors of Hsp90 with improved activities.Development of Phenyl Cyclohexylcarboxamides as a Novel Class of Hsp90 C-terminal Inhibitors.
P2860
Q35131496-FD2F7250-875C-4142-8847-F66B00E8A9C2Q35192933-17FAF450-E58D-4856-A692-8CC5BFFB2C10Q38842676-F935C328-906E-497C-828F-0173F99FF035Q39786880-271B1ACF-8A13-49CE-ACC0-E1CB3090D33DQ39867588-46362E0D-55AE-4DD8-AF30-D0AB4D8FF944Q41856020-8209B9ED-93C4-4361-89A0-ACEB027D521AQ47756540-B3575EE5-8FF8-4126-8E5F-ADA2EBE00515
P2860
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
description
2012 nî lūn-bûn
@nan
2012 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2012 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
name
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@ast
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@en
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@nl
type
label
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@ast
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@en
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@nl
prefLabel
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@ast
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@en
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues.
@nl
P2093
P2860
P356
P1476
3D-QSAR Assisted Design, Synthesis and Evaluation of Novobiocin Analogues
@en
P2093
Brian S J Blagg
Elisabetta Moroni
Huiping Zhao
P2860
P356
10.1021/ML300275G
P577
2012-01-01T00:00:00Z