Agonist derived molecular probes for A2 adenosine receptors - Wikidata - awgldk - TriplyDB

Agonist derived molecular probes for A2 adenosine receptors

Agonist derived molecular probes for A2 adenosine receptors

http://www.wikidata.org/entity/Q35170171

about

Hydrophilic side chains in the third and seventh transmembrane helical domains of human A2A adenosine receptors are required for ligand recognition 2-Substitution of N6-benzyladenosine-5'-uronamides enhances selectivity for A3 adenosine receptors Nucleoside conjugates of quantum dots for characterization of G protein-coupled receptors: strategies for immobilizing A2A adenosine receptor agonists.Functionalized congener approach to the design of ligands for G protein-coupled receptors (GPCRs).Evaluation of molecular modeling of agonist binding in light of the crystallographic structure of an agonist-bound A₂A adenosine receptor.Adenosine A1 and A2 receptors: structure--function relationships A2A adenosine receptors from rat striatum and rat pheochromocytoma PC12 cells: characterization with radioligand binding and by activation of adenylate cyclase.Behavioral effects of A1- and A2-selective adenosine agonists and antagonists: evidence for synergism and antagonism.Characterization of human striatal A2-adenosine receptors using radioligand binding and photoaffinity labeling Chemical modification and irreversible inhibition of striatal A2a adenosine receptors.Covalent binding of a selective agonist irreversibly activates guinea pig coronary artery A2 adenosine receptors.Mutagenesis reveals structure-activity parallels between human A2A adenosine receptors and biogenic amine G protein-coupled receptors.The A2 adenosine receptor: guanine nucleotide modulation of agonist binding is enhanced by proteolysis.8-(3-Chlorostyryl)caffeine (CSC) is a selective A2-adenosine antagonist in vitro and in vivo.Characterization of the locomotor depression produced by an A2-selective adenosine agonist.Fluorescent ligands for adenosine receptors.Locomotor activity in mice during chronic treatment with caffeine and withdrawal.[(3)H]XAC (xanthine amine congener) is a radioligand for A(2)-adenosine receptors in rabbit striatum.2-[2-[4-[2-[2-[ 1,3-Dihydro- 1,1-bis (4-hydroxyphenyl)-3-oxo-5-isobenzofuranthioureidyl]ethylaminocarbonyl]ethyl]phenyl] ethylamino]-5'-N-ethylcarboxamidoadenosine (FITC-APEC): A Fluorescent Ligand For A2a-Adenosine Receptors.Application of the functionalized congener approach to dendrimer-based signaling agents acting through A(2A) adenosine receptors.Adenosine A(2A) receptor dynamics studied with the novel fluorescent agonist Alexa488-APEC.

P2860

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P2860

Agonist derived molecular probes for A2 adenosine receptors

http://www.wikidata.org/entity/Q35170171

description

1989 nî lūn-bûn

@nan

1989 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած

@hyw

1989 թվականի դեկտեմբերին հրատարակված գիտական հոդված

@hy

1989年の論文

@ja

1989年論文

@yue

1989年論文

@zh-hant

1989年論文

@zh-hk

1989年論文

@zh-mo

1989年論文

@zh-tw

1989年论文

@wuu

name

Agonist derived molecular probes for A2 adenosine receptors

@ast

Agonist derived molecular probes for A2 adenosine receptors

@en

type

label

Agonist derived molecular probes for A2 adenosine receptors

@ast

Agonist derived molecular probes for A2 adenosine receptors

@en

prefLabel

Agonist derived molecular probes for A2 adenosine receptors

@ast

Agonist derived molecular probes for A2 adenosine receptors

@en

P1433

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P1476

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P2093

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P2860

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P478

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P577

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P932

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P356

P1433

Journal of Molecular Recognition

P1476

Agonist derived molecular probes for A2 adenosine receptors

@en

P2093

A J Hutchison

http://www.w3.org/2001/XMLSchema#string

G L Stiles

http://www.w3.org/2001/XMLSchema#string

K A Jacobson

http://www.w3.org/2001/XMLSchema#string

L K Pannell

http://www.w3.org/2001/XMLSchema#string

M F Jarvis

http://www.w3.org/2001/XMLSchema#string

M Williams

http://www.w3.org/2001/XMLSchema#string

W W Barrington

http://www.w3.org/2001/XMLSchema#string

X D Ji

http://www.w3.org/2001/XMLSchema#string

P2860

Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

18F-labeled insulin: a prosthetic group methodology for incorporation of a positron emitter into peptides and proteins

Electrophilic derivatives of purines as irreversible inhibitors of A1 adenosine receptors

Functionalized congeners of adenosine: preparation of analogues with high affinity for A1-adenosine receptors

High affinity acylating antagonists for the A1 adenosine receptor: identification of binding subunit

125I-labeled 8-phenylxanthine derivatives: antagonist radioligands for adenosine A1 receptors.

Identification of the A2 adenosine receptor binding subunit by photoaffinity crosslinking.

Effects of 8-phenyl and 8-cycloalkyl substituents on the activity of mono-, di-, and trisubstituted alkylxanthines with substitution at the 1-, 3-, and 7-positions.

Subclasses of external adenosine receptors.

Molecular probes for extracellular adenosine receptors.

P304

170-178

http://www.w3.org/2001/XMLSchema#string

P31

scholarly article

P356

10.1002/JMR.300020406

http://www.w3.org/2001/XMLSchema#string

P433

4

http://www.w3.org/2001/XMLSchema#string

P478

2

http://www.w3.org/2001/XMLSchema#string

P577

1989-12-01T00:00:00Z

http://www.w3.org/2001/XMLSchema#dateTime

P5875

227743528

http://www.w3.org/2001/XMLSchema#string

P698

2561548

http://www.w3.org/2001/XMLSchema#string

P932

3157953

http://www.w3.org/2001/XMLSchema#string