Structural dynamics and energetics underlying allosteric inactivation of the cannabinoid receptor CB1. - Wikidata - awgldk - TriplyDB

Structural dynamics and energetics underlying allosteric inactivation of the cannabinoid receptor CB1.

Structural dynamics and energetics underlying allosteric inactivation of the cannabinoid receptor CB1.

http://www.wikidata.org/entity/Q35845768

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Decay of an active GPCR: Conformational dynamics govern agonist rebinding and persistence of an active, yet empty, receptor state.Synthesis and biological evaluation of indole-2-carboxamides bearing photoactivatable functionalities as novel allosteric modulators for the cannabinoid CB1 receptor.Leveraging allostery to improve G protein-coupled receptor (GPCR)-directed therapeutics: cannabinoid receptor 1 as discovery target.Modulation of CB1 cannabinoid receptor by allosteric ligands: Pharmacology and therapeutic opportunities.Allosteric Modulators of the CB1 Cannabinoid Receptor: A Structural Update Review.Expression, Functional Characterization, and Solid-State NMR Investigation of the G Protein-Coupled GHS Receptor in Bilayer Membranes Biased signalling: from simple switches to allosteric microprocessors.Molecular Dynamics Methodologies for Probing Cannabinoid Ligand/Receptor Interaction.

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P2860

Structural dynamics and energetics underlying allosteric inactivation of the cannabinoid receptor CB1.

http://www.wikidata.org/entity/Q35845768

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2015 nî lūn-bûn

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Structural dynamics and energe ...... the cannabinoid receptor CB1.

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Structural dynamics and energe ...... the cannabinoid receptor CB1.

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Structural dynamics and energe ...... the cannabinoid receptor CB1.

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Structural dynamics and energe ...... the cannabinoid receptor CB1.

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Proceedings of the National Academy of Sciences of the United States of America

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Structural dynamics and energe ...... the cannabinoid receptor CB1.

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David L Farrens

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Jonathan F Fay

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P2860

Activation and allosteric modulation of a muscarinic acetylcholine receptor

Crystal structure of the β2 adrenergic receptor-Gs protein complex

Diversity and modularity of G protein-coupled receptor structures

Crystal structure of opsin in its G-protein-interacting conformation

Stabilized G protein binding site in the structure of constitutively active metarhodopsin-II

Structural Features for Functional Selectivity at Serotonin Receptors

Visualization of arrestin recruitment by a G-protein-coupled receptor

Ligand-specific endocytic dwell times control functional selectivity of the cannabinoid receptor 1

Allosteric modulation of the cannabinoid CB1 receptor

Random mutagenesis of the M3 muscarinic acetylcholine receptor expressed in yeast: identification of second-site mutations that restore function to a coupling-deficient mutant M3 receptor.

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8469-8474

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scholarly article

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27

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cannabinoid receptor

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