Reciprocal effects of an inhibitory factor on catalytic activity and noncatalytic cGMP binding sites of rod phosphodiesterase.
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Light-activated rhodopsin induces structural binding motif in G protein alpha subunitRhodopsin-transducin interface: studies with conformationally constrained peptides.Identification and characterization of a novel family of cyclic nucleotide phosphodiesterasesIsolation and characterization of a dual-substrate phosphodiesterase gene family: PDE10APhosphorylation by cyclin-dependent protein kinase 5 of the regulatory subunit of retinal cGMP phosphodiesterase. I. Identification of the kinase and its role in the turnoff of phosphodiesterase in vitro.Modulating G-protein coupled receptor/G-protein signal transduction by small molecules suggested by virtual screening.cGMP binding sites on photoreceptor phosphodiesterase: role in feedback regulation of visual transduction.Using ligand-based virtual screening to allosterically stabilize the activated state of a GPCR.Direct activation of cGMP-dependent channels of retinal rods by the cGMP phosphodiesterase.cGMP binding to noncatalytic sites on mammalian rod photoreceptor phosphodiesterase is regulated by binding of its gamma and delta subunits.cGMP is tightly bound to bovine retinal rod phosphodiesteraseBovine cone photoreceptor cGMP phosphodiesterase structure deduced from a cDNA cloneMolecular architecture of photoreceptor phosphodiesterase elucidated by chemical cross-linking and integrative modelingBinding of cGMP to the transducin-activated cGMP phosphodiesterase, PDE6, initiates a large conformational change involved in its deactivationOnset of feedback reactions underlying vertebrate rod photoreceptor light adaptationCharacterization of conformational changes and protein-protein interactions of rod photoreceptor phosphodiesterase (PDE6).Changes in cGMP concentration correlate with some, but not all, aspects of the light-regulated conductance of frog rod photoreceptorsPrenyl modification of guanine nucleotide regulatory protein gamma 2 subunits is not required for interaction with the transducin alpha subunit or rhodopsinFunctional mapping of interacting regions of the photoreceptor phosphodiesterase (PDE6) γ-subunit with PDE6 catalytic dimer, transducin, and regulator of G-protein signaling9-1 (RGS9-1).Functional exchange of components between light-activated photoreceptor phosphodiesterase and hormone-activated adenylate cyclase systemsLight-induced losses and dark recovery rates of guanosine 3',5'-cyclic monophosphate in rod outer segments of intact amphibian photoreceptors.Cone phosphodiesterase-6α' restores rod function and confers distinct physiological properties in the rod phosphodiesterase-6β-deficient rd10 mousePhosphatidylinositol-stimulated phosphorylation of an inhibitory subunit of cGMP phosphodiesterase in vertebrate rod photoreceptors.Guanosine 3',5'-cyclic nucleotide binding proteins of bovine retina identified by photoaffinity labeling.Binding of cGMP to GAF domains in amphibian rod photoreceptor cGMP phosphodiesterase (PDE). Identification of GAF domains in PDE alphabeta subunits and distinct domains in the PDE gamma subunit involved in stimulation of cGMP binding to GAF domains.Probing domain functions of chimeric PDE6alpha'/PDE5 cGMP-phosphodiesterase.Domain mapping of the retinal cyclic GMP phosphodiesterase gamma-subunit. Function of the domains encoded by the three exons of the gamma-subunit gene.Regulation of photoreceptor phosphodiesterase catalysis by its non-catalytic cGMP-binding sites.Comparison of the phosphodiesterase inhibitory subunit interactions of frog and bovine rod outer segments.Direct allosteric regulation between the GAF domain and catalytic domain of photoreceptor phosphodiesterase PDE6.Tauroursodeoxycholic acid binds to the G-protein site on light activated rhodopsin.Residues within the polycationic region of cGMP phosphodiesterase gamma subunit crucial for the interaction with transducin alpha subunit. Identification by endogenous ADP-ribosylation and site-directed mutagenesis.
P2860
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P2860
Reciprocal effects of an inhibitory factor on catalytic activity and noncatalytic cGMP binding sites of rod phosphodiesterase.
description
1982 nî lūn-bûn
@nan
1982年の論文
@ja
1982年学术文章
@wuu
1982年学术文章
@zh-cn
1982年学术文章
@zh-hans
1982年学术文章
@zh-my
1982年学术文章
@zh-sg
1982年學術文章
@yue
1982年學術文章
@zh
1982年學術文章
@zh-hant
name
Reciprocal effects of an inhib ...... ites of rod phosphodiesterase.
@ast
Reciprocal effects of an inhib ...... ites of rod phosphodiesterase.
@en
type
label
Reciprocal effects of an inhib ...... ites of rod phosphodiesterase.
@ast
Reciprocal effects of an inhib ...... ites of rod phosphodiesterase.
@en
prefLabel
Reciprocal effects of an inhib ...... ites of rod phosphodiesterase.
@ast
Reciprocal effects of an inhib ...... ites of rod phosphodiesterase.
@en
P2093
P2860
P356
P1476
Reciprocal effects of an inhib ...... ites of rod phosphodiesterase.
@en
P2093
P2860
P304
P356
10.1073/PNAS.79.12.3702
P407
P577
1982-06-01T00:00:00Z