Stimulus bias provides evidence for conformational constraints in the structure of a G protein-coupled receptor

Stimulus bias provides evidence for conformational constraints in the structure of a G protein-coupled receptor

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http://www.wikidata.org/entity/Q36347742
Non-traditional roles of G protein-coupled receptors in basic cell biologyMolecular mechanisms of bitopic ligand engagement with the M1 muscarinic acetylcholine receptorThe pharmacology of TUG-891, a potent and selective agonist of the free fatty acid receptor 4 (FFA4/GPR120), demonstrates both potential opportunity and possible challenges to therapeutic agonismEndocytic profiles of δ-opioid receptor ligands determine the duration of rapid but not sustained cAMP responses.Ligand- and cell-dependent determinants of internalization and cAMP modulation by delta opioid receptor (DOR) agonists.Mechanistic analysis of the function of agonists and allosteric modulators: reconciling two-state and operational models.Recent developments in biased agonism.Biased agonism at G protein-coupled receptors: the promise and the challenges--a medicinal chemistry perspective.Signaling within Allosteric Machines: Signal Transmission Pathways Inside G Protein-Coupled Receptors.Signaling bias in drug discovery.The mechanism of enhanced defecation caused by the ghrelin receptor agonist, ulimorelin.β2-Adrenoceptor-mediated regulation of glucose uptake in skeletal muscle--ligand-directed signalling or a reflection of system complexity?Extracellular Loop 2 of the Adenosine A1 Receptor Has a Key Role in Orthosteric Ligand Affinity and Agonist Efficacy.
P2860

Stimulus bias provides evidence for conformational constraints in the structure of a G protein-coupled receptor

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http://www.wikidata.org/entity/Q36347742
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Stimulus bias provides evidenc ...... f a G protein-coupled receptor
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Stimulus bias provides evidenc ...... f a G protein-coupled receptor
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Stimulus bias provides evidenc ...... f a G protein-coupled receptor
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Stimulus bias provides evidenc ...... f a G protein-coupled receptor
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Stimulus bias provides evidenc ...... f a G protein-coupled receptor
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Stimulus bias provides evidenc ...... f a G protein-coupled receptor
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Stimulus bias provides evidenc ...... f a G protein-coupled receptor
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P2093
P2860
P304
P31
P356
P407
P433
P478
P50
P577
P698
P921
P932