Design of 4-Oxo-1-aryl-1,4-dihydroquinoline-3-carboxamides as Selective Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 2.
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Practical Strategies and Concepts in GPCR Allosteric Modulator Discovery: Recent Advances with Metabotropic Glutamate Receptors1,3,5-Trisubstituted Pyrazoles as Potent Negative Allosteric Modulators of the mGlu2/3 Receptors.Synthesis and Preliminary Studies of a Novel Negative Allosteric Modulator, 7-((2,5-Dioxopyrrolidin-1-yl)methyl)-4-(2-fluoro-4-[11C]methoxyphenyl) quinoline-2-carboxamide, for Imaging of Metabotropic Glutamate Receptor 2.Design and Synthesis of N-Aryl Phenoxyethoxy Pyridinones as Highly Selective and CNS Penetrant mGlu3 NAMs.Design and Synthesis of mGlu2 NAMs with Improved Potency and CNS Penetration Based on a Truncated Picolinamide Core.Metabotropic glutamate receptor 2 inhibits thalamically-driven glutamate and dopamine release in the dorsal striatum.Differential Pharmacology and Binding of mGlu2 Receptor Allosteric Modulators.
P2860
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P2860
Design of 4-Oxo-1-aryl-1,4-dihydroquinoline-3-carboxamides as Selective Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 2.
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2015 nî lūn-bûn
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2015年の論文
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2015年論文
@yue
2015年論文
@zh-hant
2015年論文
@zh-hk
2015年論文
@zh-mo
2015年論文
@zh-tw
2015年论文
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2015年论文
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2015年论文
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name
Design of 4-Oxo-1-aryl-1,4-dih ...... Glutamate Receptor Subtype 2.
@ast
Design of 4-Oxo-1-aryl-1,4-dih ...... Glutamate Receptor Subtype 2.
@en
type
label
Design of 4-Oxo-1-aryl-1,4-dih ...... Glutamate Receptor Subtype 2.
@ast
Design of 4-Oxo-1-aryl-1,4-dih ...... Glutamate Receptor Subtype 2.
@en
prefLabel
Design of 4-Oxo-1-aryl-1,4-dih ...... Glutamate Receptor Subtype 2.
@ast
Design of 4-Oxo-1-aryl-1,4-dih ...... Glutamate Receptor Subtype 2.
@en
P2093
P2860
P50
P1476
Design of 4-Oxo-1-aryl-1,4-dih ...... Glutamate Receptor Subtype 2.
@en
P2093
Alice L Rodriguez
Andrew S Felts
Anna L Blobaum
Charles W Locuson
Daryl F Venable
Frank W Byers
J Scott Daniels
Julie L Engers
Katrina A Smith
Kyle A Emmitte
P2860
P304
P356
10.1021/ACS.JMEDCHEM.5B01371
P407
P577
2015-11-02T00:00:00Z