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Designing the next generation of medicines for malaria control and eradicationMalaria in South America: a drug discovery perspectiveA chemical proteomics approach for the search of pharmacological targets of the antimalarial clinical candidate albitiazolium in Plasmodium falciparum using photocrosslinking and click chemistryA Divergent SAR Study Allows Optimization of a Potent 5-HT2c Inhibitor to a Promising Antimalarial Scaffold.Screening and hit evaluation of a chemical library against blood-stage Plasmodium falciparum.Antimalarial aminothiazoles and aminopyridines from phenotypic whole-cell screening of a SoftFocus(®) library.Whole-cell in vitro screening for gametocytocidal compounds.Drug repositioning as a route to anti-malarial drug discovery: preliminary investigation of the in vitro anti-malarial efficacy of emetine dihydrochloride hydrate.Nowhere to hide: interrogating different metabolic parameters of Plasmodium falciparum gametocytes in a transmission blocking drug discovery pipeline towards malaria elimination.Inclusion of gametocyte parameters in anti-malarial drug efficacy studies: filling a neglected gap needed for malaria eliminationA framework for assessing the risk of resistance for anti-malarials in development.Sustainable malaria control: transdisciplinary approaches for translational applications.Anthracene-polyamine conjugates inhibit in vitro proliferation of intraerythrocytic Plasmodium falciparum parasitesSynthesis of a potent antimalarial agent through natural products conjugation.Fast in vitro methods to determine the speed of action and the stage-specificity of anti-malarials in Plasmodium falciparum.Antimalarial drug discovery - the path towards eradication.New approaches in antimalarial drug discovery and development: a review.Role of Different Pfcrt and Pfmdr-1 Mutations in Conferring Resistance to Antimalaria Drugs in Plasmodium falciparum.Resisting resistance: is there a solution for malaria?Case Study of Small Molecules As Antimalarials: 2-Amino-1-phenylethanol (APE) Derivatives.Evaluation of bioluminescence-based assays of anti-malarial drug activity.Stoking the drug target pipeline for human African trypanosomiasis.A global survey of ATPase activity in Plasmodium falciparum asexual blood stages and gametocytes.Antimalarial drug discovery: where next?Isolation and synthesis of falcitidin, a novel myxobacterial-derived acyltetrapeptide with activity against the malaria target falcipain-2.Interview with Future Medicinal Chemistry's US Senior Editor, Iwao Ojima. Interview by Issac Bruce.Drugs for neglected diseases: part II.The role of modern drug discovery in the fight against neglected and tropical diseases
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description
article científic
@ca
article scientifique
@fr
articol științific
@ro
articolo scientifico
@it
artigo científico
@gl
artigo científico
@pt
artigo científico
@pt-br
artikel ilmiah
@id
artikull shkencor
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artículo científico
@es
name
Challenges in antimalarial drug discovery.
@en
Challenges in antimalarial drug discovery.
@nl
type
label
Challenges in antimalarial drug discovery.
@en
Challenges in antimalarial drug discovery.
@nl
prefLabel
Challenges in antimalarial drug discovery.
@en
Challenges in antimalarial drug discovery.
@nl
P2093
P2860
P356
P1476
Challenges in antimalarial drug discovery.
@en
P2093
David Waterson
Didier Leroy
Julie Lotharius
P2860
P304
P356
10.4155/FMC.11.91
P577
2011-09-01T00:00:00Z