New modalities in conformationally constrained peptides for potency, selectivity and cell permeation.
about
Racemic and quasi-racemic X-ray structures of cyclic disulfide-rich peptide drug scaffoldsNeighbor-directed histidine N (τ)-alkylation: A route to imidazolium-containing phosphopeptide macrocyclesConstraining cyclic peptides to mimic protein structure motifs.Comparative α-helicity of cyclic pentapeptides in water.Cone snail venomics: from novel biology to novel therapeutics.Stapled Peptides by Late-Stage C(sp3 )-H Activation.Strategies to stabilize cell penetrating peptides for in vivo applications.Direct targeting of Rab-GTPase-effector interactions.Synthesis of bioactive and stabilized cyclic peptides by macrocyclization using C(sp3)-H activation.Cathelicidin-trypsin inhibitor loop conjugate represents a promising antibiotic candidate with protease stabilityNew peptide architectures through C-H activation stapling between tryptophan-phenylalanine/tyrosine residuesConstrained Cyclopeptides: Biaryl Formation through Pd-Catalyzed C-H Activation in Peptides-Structural Control of the Cyclization vs. Cyclodimerization Outcome.Design, synthesis, and opioid activity of arodyn analogs cyclized by ring-closing metathesis involving Tyr(allyl).Stapled Peptides by Late-Stage C(sp3)−H ActivationComparison of hydrocarbon-and lactam-bridged cyclic peptides as dimerization inhibitors of Leishmania infantum trypanothione reductase
P2860
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P2860
New modalities in conformationally constrained peptides for potency, selectivity and cell permeation.
description
article científic
@ca
article scientifique
@fr
articol științific
@ro
articolo scientifico
@it
artigo científico
@gl
artigo científico
@pt
artigo científico
@pt-br
artikel ilmiah
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artikull shkencor
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artículo científico
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name
New modalities in conformation ...... lectivity and cell permeation.
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type
label
New modalities in conformation ...... lectivity and cell permeation.
@en
prefLabel
New modalities in conformation ...... lectivity and cell permeation.
@en
P2860
P356
P1476
New modalities in conformation ...... lectivity and cell permeation.
@en
P2093
Ram Dharanipragada
P2860
P304
P356
10.4155/FMC.13.25
P577
2013-05-01T00:00:00Z