Structure-activity relationships and mechanism of action of Eph-ephrin antagonists: interaction of cholanic acid with the EphA2 receptor.
about
Discovery of a Novel Chemotype of Tyrosine Kinase Inhibitors by Fragment-Based Docking and Molecular DynamicsInhibition of Eph receptor-ephrin ligand interaction by tea polyphenols.UniPR129 is a competitive small molecule Eph-ephrin antagonist blocking in vitro angiogenesis at low micromolar concentrations.Comparative Analysis of Virtual Screening Approaches in the Search for Novel EphA2 Receptor Antagonists.Steroids as γ-secretase modulators.Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor.Synthesis and structure-activity relationships of amino acid conjugates of cholanic acid as antagonists of the EphA2 receptor.Target hopping as a useful tool for the identification of novel EphA2 protein-protein antagonists.Fluorine-18 radiolabeling and radiopharmacological characterization of a benzodioxolylpyrimidine-based radiotracer targeting the receptor tyrosine kinase EphB4.Design, synthesis and characterization of novel small molecular inhibitors of ephrin-B2 binding to EphB4.An efficient bioorthogonal strategy using CuAAC click chemistry for radiofluorinations of SNEW peptides and the role of copper depletion.Exploiting Free-Energy Minima to Design Novel EphA2 Protein-Protein Antagonists: From Simulation to Experiment and Return.
P2860
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P2860
Structure-activity relationships and mechanism of action of Eph-ephrin antagonists: interaction of cholanic acid with the EphA2 receptor.
description
2012 nî lūn-bûn
@nan
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
2012年论文
@zh
2012年论文
@zh-cn
name
Structure-activity relationshi ...... acid with the EphA2 receptor.
@en
Structure-activity relationshi ...... acid with the EphA2 receptor.
@nl
type
label
Structure-activity relationshi ...... acid with the EphA2 receptor.
@en
Structure-activity relationshi ...... acid with the EphA2 receptor.
@nl
prefLabel
Structure-activity relationshi ...... acid with the EphA2 receptor.
@en
Structure-activity relationshi ...... acid with the EphA2 receptor.
@nl
P2093
P2860
P356
P1433
P1476
Structure-activity relationshi ...... acid with the EphA2 receptor.
@en
P2093
Alessio Lodola
Barbara Lelli
Carmine Giorgio
Elena B Pasquale
Elisabetta Barocelli
Iftiin Hassan-Mohamed
Luisa Bracci
Massimiliano Tognolini
Matteo Incerti
P2860
P304
P356
10.1002/CMDC.201200102
P577
2012-04-23T00:00:00Z