Solid phase synthesis and structural analysis of novel A-chain dicarba analogs of human relaxin-3 (INSL7) that exhibit full biological activity.

Solid phase synthesis and structural analysis of novel A-chain dicarba analogs of human relaxin-3 (INSL7) that exhibit full biological activity.

Item
http://www.wikidata.org/entity/Q39864557
Synthesis of chemically modified bioactive peptides: recent advances, challenges and developments for medicinal chemistry.Synthetic covalently linked dimeric form of H2 relaxin retains native RXFP1 activity and has improved in vitro serum stability.The minimal active structure of human relaxin-2The different ligand-binding modes of relaxin family peptide receptors RXFP1 and RXFP2Peptides and proteins as a continuing exciting source of inspiration for peptidomimetics.Microwave heating in solid-phase peptide synthesis.Total Chemical Synthesis of an Intra-A-Chain Cystathionine Human Insulin Analogue with Enhanced Thermal Stability.Synthesis, conformational analysis and biological properties of a dicarba derivative of the antimicrobial peptide, brevinin-1BYa.Chemically synthesized dicarba H2 relaxin analogues retain strong RXFP1 receptor activity but show an unexpected loss of in vitro serum stability.Total chemical synthesis of a heterodimeric interchain bis-lactam-linked Peptide: application to an analogue of human insulin-like Peptide 3.Insulin in motion: The A6-A11 disulfide bond allosterically modulates structural transitions required for insulin activity.Disulfide Bond Mimetics: Strategies and Challenges.Diaminodiacid Bridges to Improve Folding and Tune the Bioactivity of Disulfide-Rich Peptides.Urotensin-II peptidomimetic incorporating a non-reducible 1,5-triazole disulfide bond reveals a pseudo-irreversible covalent binding mechanism to the urotensin G-protein coupled receptor.
P2860

Solid phase synthesis and structural analysis of novel A-chain dicarba analogs of human relaxin-3 (INSL7) that exhibit full biological activity.

Item
http://www.wikidata.org/entity/Q39864557
description
2009 nî lūn-bûn
@nan
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
2009年论文
@zh
2009年论文
@zh-cn
name
Solid phase synthesis and stru ...... ibit full biological activity.
@en
Solid phase synthesis and stru ...... rba analogs of human relaxin-3
@nl
type
label
Solid phase synthesis and stru ...... ibit full biological activity.
@en
Solid phase synthesis and stru ...... rba analogs of human relaxin-3
@nl
prefLabel
Solid phase synthesis and stru ...... ibit full biological activity.
@en
Solid phase synthesis and stru ...... rba analogs of human relaxin-3
@nl
P1433
P1476
P2093
P2860
P304
P31
P356
P433
P478
P50
P577
P5875
P698
P356
P1433
P1476
Solid phase synthesis and stru ...... ibit full biological activity.
@en
P2093
P2860
P304
P31
P356
P433
P478
P50
P577
P5875
P698